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Compound Detail

CHEMBL489380

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O=C1Nc2ccc(OC(F)(F)F)cc2/C1=N/NC(=S)Nc1ccccc1

Basic Information

ChEMBL ID CHEMBL489380
Phase Preclinical
Structure Type MOL
InChI Key WHVILFJSEYISRF-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

380.4
MW (Da)
3.23
ALogP
4
HBA
3
HBD
74.8
PSA (Ų)
0.56
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H11F3N4O2S
MW 380.35
Aromatic Rings 2
Heavy Atoms 26
NP-Likeness -1.65

Activity Summary

IC50 1 meas. best 5.23

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human alphaherpesvirus 1
CHEMBL377
IC50 5.23 5.23 5900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Human alphaherpesvirus 1 IC50 = 5900.0 nM 5.23 Antiviral activity against HSV1 by plaque reduction assay 21356589

Literature References

PubMed DOI Target Context # Activities
18804379 10.1016/j.bmc.2008.08.050 Mycobacterium tuberculosis 1
18804379 10.1016/j.bmc.2008.08.050 Vero 1
21356589 10.1016/j.bmcl.2011.02.037 Human alphaherpesvirus 1 1
21356589 10.1016/j.bmcl.2011.02.037 Human alphaherpesvirus 2 1
21356589 10.1016/j.bmcl.2011.02.037 RD 1

Data from ChEMBL 36 via Core Engine