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Compound Detail

CHEMBL505662

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CCCCCCCCC1(CCCCCCCC)O[C@H]2[C@H](OC(=O)/C=C/c3ccc(O)c(O)c3)C[C@]3(C[C@H]2O1)OC(CCCCCCCC)(CCCCCCCC)OC3=O

Basic Information

ChEMBL ID CHEMBL505662
Phase Preclinical
Structure Type MOL
InChI Key RODCZSHMCGJEBO-LHWIJXPWSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

827.2
MW (Da)
13.31
ALogP
9
HBA
2
HBD
120.8
PSA (Ų)
0.03
QED
2
Ro5 Violations
31
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C50H82O9
MW 827.20
Aromatic Rings 1
Heavy Atoms 59
NP-Likeness 0.75

Activity Summary

IC50 2 meas. best 6.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.3 6.175 500.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
18783210 10.1021/jm800621x Unchecked 2

Data from ChEMBL 36 via Core Engine