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Compound Detail

CHEMBL506444

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CCC1(N)C2CC3CC(C2)CC1C3.Cl

Basic Information

ChEMBL ID CHEMBL506444
Phase Preclinical
Structure Type MOL
InChI Key JKDUTNHREIIDCM-UHFFFAOYSA-N
Parent Compound CHEMBL1170181
Active Moiety CHEMBL1170181
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
5
Publications
0
Known Names

Molecular Properties

179.3
MW (Da)
2.55
ALogP
1
HBA
1
HBD
26.0
PSA (Ų)
0.66
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C12H22ClN
MW 215.77
Aromatic Rings 0
Heavy Atoms 13
NP-Likeness 0.84

Activity Summary

Kd 1 meas. best 5.17

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Kd 5.17 5.17 6700.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked Kd = 6700.0 nM 5.17 Binding affinity to influenza A virus A/chicken/Germany/27 H7N7 weybridge strain... 18947998

Literature References

PubMed DOI Target Context # Activities
18947998 10.1016/j.bmcl.2008.10.003 Unchecked 1
18947998 10.1016/j.bmcl.2008.10.003 H2N2 subtype 1
18947998 10.1016/j.bmcl.2008.10.003 Influenza A virus 1
18947998 10.1016/j.bmcl.2008.10.003 Influenza B virus 1
18947998 10.1016/j.bmcl.2008.10.003 MDCK 1

Data from ChEMBL 36 via Core Engine