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Compound Detail

CHEMBL5080591

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OCC[N+]1(CCCCCCOc2ccc(C(=C3C4CC5CC(C4)CC3C5)c3ccc(OCCCCCC[N+]4(CCO)CCCC4)cc3)cc2)CCCC1.[I-].[I-]

Basic Information

ChEMBL ID CHEMBL5080591
Phase Preclinical
Structure Type MOL
InChI Key COPRQIADRSNKOB-UHFFFAOYSA-L
Parent Compound CHEMBL5095626
Active Moiety CHEMBL5095626
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

729.1
MW (Da)
9.03
ALogP
4
HBA
2
HBD
58.9
PSA (Ų)
0.09
QED
2
Ro5 Violations
22
Rot. Bonds

Drug Information

Molecule Type Unknown
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C47H72I2N2O4
MW 982.91
Aromatic Rings 2
Heavy Atoms 53
NP-Likeness 0.02

Activity Summary

IC50 1 meas. best 5.8

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
MCF7
CHEMBL387
IC50 5.8 5.8 1600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
MCF7 IC50 = 1600.0 nM 5.8 Antiproliferative activity against human MCF7 cells measured by WST-1 assay -

Data from ChEMBL 36 via Core Engine