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Compound Detail

CHEMBL517681

METHYLINOSCAVIN A
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COc1cc(/C=C/c2cc3c(c(=O)o2)C2(OC(C)=CC2=O)C(c2ccc(O)c(O)c2)O3)ccc1O

Basic Information

ChEMBL ID CHEMBL517681
Name METHYLINOSCAVIN A
Phase Preclinical
Structure Type MOL
InChI Key LNCIAIFVVJWMRV-ZZXKWVIFSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

476.4
MW (Da)
3.77
ALogP
9
HBA
3
HBD
135.7
PSA (Ų)
0.48
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C26H20O9
MW 476.44
Aromatic Rings 3
Heavy Atoms 35
NP-Likeness 1.78

Activity Summary

IC50 2 meas. best 4.97

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 4.97 4.835 10700.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
16499338 10.1021/np050453n NON-PROTEIN TARGET 2
16499338 10.1021/np050453n Radical scavenging activity 1

Data from ChEMBL 36 via Core Engine