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Compound Detail

CHEMBL517790

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C[C@H]1C[C@H]([C@](C)(O)[C@H]2CC[C@H]3[C@@H]4C[C@H]5O[C@]56[C@@H](O)C=CC(=O)[C@]6(C)[C@H]4CC[C@]23C)OC(=O)[C@@H]1C

Basic Information

ChEMBL ID CHEMBL517790
Phase Preclinical
Structure Type MOL
InChI Key OGABYGZTMRAASL-UWCCFGPMSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

472.6
MW (Da)
3.43
ALogP
6
HBA
2
HBD
96.4
PSA (Ų)
0.47
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C28H40O6
MW 472.62
Aromatic Rings 0
Heavy Atoms 34
NP-Likeness 3.73

Activity Summary

IC50 1 meas. best 5.26

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
ADMET
CHEMBL612558
IC50 5.26 5.26 5500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
ADMET IC50 = 5500.0 nM 5.26 Growth inhibition of mouse Hepa-1c1c7 cells by crystal violet staining 12027740

Literature References

PubMed DOI Target Context # Activities
12027740 10.1021/np0106337 Quinone oxidoreductase 2
12027740 10.1021/np0106337 Unchecked 2
12027740 10.1021/np0106337 ADMET 1

Data from ChEMBL 36 via Core Engine