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Compound Detail

CHEMBL5178531

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COc1cc([C@@H]2c3c(O)cc(O)cc3[C@@H]3[C@H]2CO[C@H]3c2cc(O)c(O)c(O)c2)cc(OC)c1O

Basic Information

ChEMBL ID CHEMBL5178531
Phase Preclinical
Structure Type MOL
InChI Key UNFKSXAIQDLCLW-KWTWETESSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

468.5
MW (Da)
3.55
ALogP
9
HBA
6
HBD
149.1
PSA (Ų)
0.32
QED
1
Ro5 Violations
4
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C25H24O9
MW 468.46
Aromatic Rings 3
Heavy Atoms 34
NP-Likeness 1.66

Activity Summary

IC50 1 meas. best 5.19

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.19 5.19 6500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 6500.0 nM 5.19 Inhibition of Bacillus stearothermophilus alpha-glucosidase type IV using p-nitr... 35367706

Literature References

PubMed DOI Target Context # Activities
35367706 10.1016/j.ejmech.2022.114282 Unchecked 1

Data from ChEMBL 36 via Core Engine