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Compound Detail

CHEMBL518101

BROUSSOCHALCONE TRIACETATE
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CC(=O)Oc1cc(O)c(C(=O)/C=C/c2ccc(OC(C)=O)c(OC(C)=O)c2)cc1CC=C(C)C

Basic Information

ChEMBL ID CHEMBL518101
Name BROUSSOCHALCONE TRIACETATE
Phase Preclinical
Structure Type MOL
InChI Key OSMAHDXNHPCYBB-JXMROGBWSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

466.5
MW (Da)
4.57
ALogP
8
HBA
1
HBD
116.2
PSA (Ų)
0.20
QED
0
Ro5 Violations
8
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C26H26O8
MW 466.49
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness 0.97

Activity Summary

IC50 1 meas. best 4.04

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
NON-PROTEIN TARGET
CHEMBL3879801
IC50 4.04 4.04 91700.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
NON-PROTEIN TARGET IC50 = 91700.0 nM 4.04 Antiplatelet activity against rabbit platelets assessed as arachidonic acid-indu... 8864236

Literature References

PubMed DOI Target Context # Activities
8864236 10.1021/np960376j NON-PROTEIN TARGET 9

Data from ChEMBL 36 via Core Engine