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Compound Detail

CHEMBL5206488

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COC(=O)c1ccc(C(=O)NNc2c(Br)cccc2Br)cc1

Basic Information

ChEMBL ID CHEMBL5206488
Phase Preclinical
Structure Type MOL
InChI Key KKQWVAZLYCVAGY-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

428.1
MW (Da)
3.76
ALogP
4
HBA
2
HBD
67.4
PSA (Ų)
0.58
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C15H12Br2N2O3
MW 428.08
Aromatic Rings 2
Heavy Atoms 22
NP-Likeness -0.95

Activity Summary

EC50 1 meas. best 6.48

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Influenza A virus
CHEMBL613740
EC50 6.48 6.48 330.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Influenza A virus EC50 = 330.0 nM 6.48 Antiviral activity against influenza A virus H5N1 infected in dog MDCK cells ass... 35212527

Literature References

PubMed DOI Target Context # Activities
35212527 10.1021/acs.jmedchem.1c01257 Influenza A virus 1
35212527 10.1021/acs.jmedchem.1c01257 MDCK 1
35212527 10.1021/acs.jmedchem.1c01257 ADMET 1

Data from ChEMBL 36 via Core Engine