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Compound Detail

CHEMBL52271

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C=CCSCc1c(O)c(CSCC=C)c2c(c1O)C[C@@H](OC(=O)c1cc(O)c(O)c(O)c1)[C@@H](c1cc(O)c(O)c(O)c1)O2

Basic Information

ChEMBL ID CHEMBL52271
Phase Preclinical
Structure Type MOL
InChI Key NMTWEDAQPKKZDB-QDPGVEIFSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

630.7
MW (Da)
5.07
ALogP
13
HBA
8
HBD
197.4
PSA (Ų)
0.06
QED
4
Ro5 Violations
11
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C30H30O11S2
MW 630.69
Aromatic Rings 3
Heavy Atoms 43
NP-Likeness 1.14

Activity Summary

IC50 1 meas. best 4.94

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.94 4.94 11600.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 11600.0 nM 4.94 Inhibitory activity against lipid peroxidation of egg-phosphatidylcholine (PC) l... 9873437

Literature References

PubMed DOI Target Context # Activities
9873437 10.1016/s0960-894x(98)00311-4 Unchecked 2
9873437 10.1016/s0960-894x(98)00311-4 No relevant target 1

Data from ChEMBL 36 via Core Engine