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Compound Detail

CHEMBL52561

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CCCCCCCCCCCCCCCCCCNC(=O)Oc1c(O)cc(C(=O)O[C@@H]2Cc3c(O)cc(O)cc3O[C@@H]2c2cc(O)c(O)c(O)c2)cc1O

Basic Information

ChEMBL ID CHEMBL52561
Phase Preclinical
Structure Type MOL
InChI Key SNRYCHOAZPOTPP-XXKIVBBDSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

753.9
MW (Da)
8.88
ALogP
12
HBA
8
HBD
215.5
PSA (Ų)
0.03
QED
4
Ro5 Violations
21
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C41H55NO12
MW 753.89
Aromatic Rings 3
Heavy Atoms 54
NP-Likeness 1.05

Activity Summary

IC50 2 meas. best 4.66

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.66 4.635 22100.0 2

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
9873437 10.1016/s0960-894x(98)00311-4 Unchecked 2
9873437 10.1016/s0960-894x(98)00311-4 No relevant target 1

Data from ChEMBL 36 via Core Engine