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Compound Detail

CHEMBL541380

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CCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCCCCNCC.Cl

Basic Information

ChEMBL ID CHEMBL541380
Phase Preclinical
Structure Type MOL
InChI Key AGLLDILTWGINCP-UHFFFAOYSA-N
Parent Compound CHEMBL1190697
Active Moiety CHEMBL1190697
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

997.7
MW (Da)
5.42
ALogP
14
HBA
14
HBD
168.4
PSA (Ų)
0.03
QED
4
Ro5 Violations
67
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C56H129ClN14
MW 1034.20
Aromatic Rings 0
Heavy Atoms 70
NP-Likeness -0.02

Activity Summary

EC50 1 meas. best 5.05

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Leishmania donovani
CHEMBL367
EC50 5.05 5.05 9000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Leishmania donovani EC50 = 9000.0 nM 5.05 Antiproliferative activity against Leishmania donovani DI700 promastigotes 17116678

Literature References

PubMed DOI Target Context # Activities
17116678 10.1128/aac.01193-06 Leishmania donovani 2

Data from ChEMBL 36 via Core Engine