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Compound Detail

CHEMBL550359

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O=C(N[C@@H]1CCCc2c1[nH]c1ccc(Cl)cc21)c1ccccc1F

Basic Information

ChEMBL ID CHEMBL550359
Phase Preclinical
Structure Type MOL
InChI Key TXFFKXTVYMUXME-QGZVFWFLSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
4
Publications
0
Known Names

Molecular Properties

342.8
MW (Da)
4.77
ALogP
1
HBA
2
HBD
44.9
PSA (Ų)
0.69
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H16ClFN2O
MW 342.80
Aromatic Rings 3
Heavy Atoms 24
NP-Likeness -1.20

Activity Summary

IC50 1 meas. best 8.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Human papillomavirus type 16
CHEMBL613205
IC50 8.1 8.1 8.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
19556128 10.1016/j.bmcl.2009.06.001 Human papillomavirus type 16 1
19556128 10.1016/j.bmcl.2009.06.001 HFF 1
19556128 10.1016/j.bmcl.2009.06.001 Cytochrome P450 2D6 1
19556128 10.1016/j.bmcl.2009.06.001 Voltage-gated inwardly rectifying potassium channel KCNH2 1

Data from ChEMBL 36 via Core Engine