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Compound Detail

CHEMBL557703

SOPHONOROL C
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COc1c([C@]2(O)COc3c4c(cc(O)c3C2=O)OC(C)(C)CC4)ccc2c1CCC(C)(C)O2

Basic Information

ChEMBL ID CHEMBL557703
Name SOPHONOROL C
Phase Preclinical
Structure Type MOL
InChI Key VTNVBSWKRFKHFA-AREMUKBSSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
2
Publications
0
Known Names

Molecular Properties

454.5
MW (Da)
4.07
ALogP
7
HBA
2
HBD
94.5
PSA (Ų)
0.71
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C26H30O7
MW 454.52
Aromatic Rings 2
Heavy Atoms 33
NP-Likeness 1.86

Activity Summary

IC50 1 meas. best 4.89

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Plasmodium falciparum
CHEMBL364
IC50 4.89 4.89 12900.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Plasmodium falciparum IC50 = 12900.0 nM 4.89 Antiplasmodial activity against chloroquine-sensitive Plasmodium falciparum D10 19572738

Literature References

PubMed DOI Target Context # Activities
19572738 10.1021/np900144c Plasmodium falciparum 1
19572738 10.1021/np900144c CHO 1

Data from ChEMBL 36 via Core Engine