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Compound Detail

CHEMBL558301

SOPHONOROL F
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COc1cc(O)c2c(c1CC=C(C)C)OC[C@@](O)(c1ccc(O)c(CC=C(C)C)c1OC)C2=O

Basic Information

ChEMBL ID CHEMBL558301
Name SOPHONOROL F
Phase Preclinical
Structure Type MOL
InChI Key CXAXZPWQRPXPGL-HHHXNRCGSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

468.6
MW (Da)
4.60
ALogP
7
HBA
3
HBD
105.5
PSA (Ų)
0.51
QED
0
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C27H32O7
MW 468.55
Aromatic Rings 2
Heavy Atoms 34
NP-Likeness 2.05

Activity Summary

IC50 2 meas. best 4.39

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Plasmodium falciparum
CHEMBL364
IC50 4.39 4.39 41000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Plasmodium falciparum IC50 = 41000.0 nM 4.39 Antiplasmodial activity against chloroquine-sensitive Plasmodium falciparum D10 19572738

Literature References

PubMed DOI Target Context # Activities
19572738 10.1021/np900144c Plasmodium falciparum 1
19572738 10.1021/np900144c CHO 1
19572738 10.1021/np900144c Unchecked 1

Data from ChEMBL 36 via Core Engine