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Compound Detail

CHEMBL5593882

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Cc1cc(C)cc(N2C(=O)C[n+]3ccccc3C2C(=O)Nc2ccc(Cl)cc2)c1

Basic Information

ChEMBL ID CHEMBL5593882
Phase Preclinical
Structure Type MOL
InChI Key QJKQDAKMOLOLGR-UHFFFAOYSA-O
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

406.9
MW (Da)
3.97
ALogP
2
HBA
1
HBD
53.3
PSA (Ų)
0.67
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H21ClN3O2+
MW 406.89
Aromatic Rings 3
Heavy Atoms 29
NP-Likeness -1.12

Activity Summary

IC50 1 meas. best 5.06

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Replicase polyprotein 1ab
CHEMBL4523582
IC50 5.06 5.06 8800.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Replicase polyprotein 1ab IC50 = 8800.0 nM 5.06 Inhibition of SARS CoV-2 main protease 37944867

Literature References

PubMed DOI Target Context # Activities
37944867 10.1016/j.bmcl.2023.129547 Replicase polyprotein 1ab 2

Data from ChEMBL 36 via Core Engine