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Compound Detail

CHEMBL565816

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CCCCCCCCCCCCCCCCCC(=O)N(C)C[C@@H](O)COP(=O)(O)OC[C@H](N)C(=O)O

Basic Information

ChEMBL ID CHEMBL565816
Phase Preclinical
Structure Type MOL
InChI Key NOHULNIVDHURHZ-PKTZIBPZSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

538.7
MW (Da)
4.61
ALogP
7
HBA
4
HBD
159.6
PSA (Ų)
0.10
QED
1
Ro5 Violations
25
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C25H51N2O8P
MW 538.66
Aromatic Rings 0
Heavy Atoms 36
NP-Likeness 0.18

Activity Summary

EC50 1 meas. best 5.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Mast cell
CHEMBL613709
EC50 5.0 5.0 10000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Mast cell EC50 = 10000.0 nM 5.0 Induction of Wistar rat peritoneal mast cell degradation assessed as concanavali... 19743861

Literature References

PubMed DOI Target Context # Activities
19743861 10.1021/jm900598m Mast cell 4

Data from ChEMBL 36 via Core Engine