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Compound Detail

CHEMBL56686

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C=C1/C(=C\C=C2/CCC[C@@]3(C)C2CC[C@@H]3[C@H](C)/C=C/C(C)C(C)(O)CO)C[C@@H](O)C[C@@H]1O

Basic Information

ChEMBL ID CHEMBL56686
Phase Preclinical
Structure Type MOL
InChI Key BXQJQHRLBLTYMC-YTMNFUGOSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

444.7
MW (Da)
4.70
ALogP
4
HBA
4
HBD
80.9
PSA (Ų)
0.45
QED
0
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C28H44O4
MW 444.66
Aromatic Rings 0
Heavy Atoms 32
NP-Likeness 2.60

Activity Summary

IC50 1 meas. best 8.1

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
RWLeu4
CHEMBL614885
IC50 8.1 8.1 8.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
RWLeu4 IC50 = 8.0 nM 8.1 Concentration required to decrease [3H]thymidine incorporation by 50 percent in ... -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(00)80123-7 RWLeu4 4

Data from ChEMBL 36 via Core Engine