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Compound Detail

CHEMBL5790440

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CN(C)c1ccc(C#Cc2cc3ccc(-c4ccsc4)nc3[nH]2)cc1

Basic Information

ChEMBL ID CHEMBL5790440
Phase Preclinical
Structure Type MOL
InChI Key SPYYWCDGZNJHNH-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

343.4
MW (Da)
4.76
ALogP
3
HBA
1
HBD
31.9
PSA (Ų)
0.53
QED
0
Ro5 Violations
2
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H17N3S
MW 343.45
Aromatic Rings 4
Heavy Atoms 25
NP-Likeness -1.52

Activity Summary

Kd 2 meas. best 9.14

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Alpha-synuclein
CHEMBL6152
Kd 9.14 9.14 0.7 1
Unchecked
CHEMBL612545
Kd 8.37 8.37 4.3 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine