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Compound Detail

CHEMBL5808975

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CCOC(=O)/C(C)=C/c1cc(F)c(Oc2ccc(S(=O)(=O)NCCOCCOCCOCCOCCOCCOCCN)cc2)c(F)c1

Basic Information

ChEMBL ID CHEMBL5808975
Phase Preclinical
Structure Type MOL
InChI Key CGGLCPZFGSPZFV-YYDJUVGSSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

704.8
MW (Da)
3.06
ALogP
12
HBA
2
HBD
163.1
PSA (Ų)
0.08
QED
2
Ro5 Violations
27
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C32H46F2N2O11S
MW 704.79
Aromatic Rings 2
Heavy Atoms 48
NP-Likeness -0.51

Activity Summary

IC50 1 meas. best 6.5

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 6.5 6.5 316.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 316.0 nM 6.5 Cell-Based Assay of NHE-3 Activity: Rat NHE-3-mediated Na+-dependent H+ antiport... -

Data from ChEMBL 36 via Core Engine