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Compound Detail

CHEMBL5826590

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Cn1cc(-c2cn[nH]c2)c2cc(C#CC3(O)CCCC3)ncc21

Basic Information

ChEMBL ID CHEMBL5826590
Phase Preclinical
Structure Type MOL
InChI Key IFNZGRFIBOXNAH-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

306.4
MW (Da)
2.62
ALogP
4
HBA
2
HBD
66.7
PSA (Ų)
0.68
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C18H18N4O
MW 306.37
Aromatic Rings 3
Heavy Atoms 23
NP-Likeness -0.42

Activity Summary

IC50 1 meas. best 7.68

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Inhibitor of nuclear factor kappa-B kinase subunit alpha
CHEMBL3476
IC50 7.68 7.68 21.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine