Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL5830357

Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
COc1cc(N[C+](C(=O)N2CCc3ccc(S(F)(F)(F)(F)F)cc32)c2ccc(Cl)cc2)cc(OCCCC(=O)O)c1

Basic Information

ChEMBL ID CHEMBL5830357
Phase Preclinical
Structure Type MOL
InChI Key WOHNQOKYAYUIPX-UHFFFAOYSA-O
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

620.0
MW (Da)
7.83
ALogP
5
HBA
2
HBD
88.1
PSA (Ų)
0.13
QED
2
Ro5 Violations
11
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C27H25ClF5N2O5S+
MW 620.02
Aromatic Rings 3
Heavy Atoms 41
NP-Likeness -0.54

Activity Summary

EC50 1 meas. best 9.96

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Genome polyprotein
CHEMBL5980
EC50 9.96 9.96 0.1 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Genome polyprotein EC50 = 0.11 nM 9.96 DENV-2 Antiviral Assay: The antiviral activity of all the compounds of the inven... -

Data from ChEMBL 36 via Core Engine