Skip to main content
Free research Free research Free compound review with research home and workspace preview
Quick search ChEMBL 36
Compound Detail

CHEMBL5940975

RG6341
🧪 Phase II
Enter ChEMBL ID:
Free Research Context This compound will appear in recent viewed items on the research home for this browser.
Research home View demo workspace
🧪 Phase II
Cc1nc2ncn(C)c2c(=O)n1Cc1nc([C@@H]2CO[C@@H](c3ccc(Cl)cc3)C2)no1

Basic Information

ChEMBL ID CHEMBL5940975
Name RG6341
Phase Phase II
Structure Type MOL
InChI Key FIBJEOLUMVIRIT-DZGCQCFKSA-N

Known Names

Gdc-6599 Rg-6341 Rg6341
1
Targets
4
Activities
1
Assay Types
0
PK Parameters
0
Publications
3
Known Names

Molecular Properties

426.9
MW (Da)
2.77
ALogP
9
HBA
0
HBD
100.9
PSA (Ų)
0.49
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Chirality Single Enantiomer

Extended Properties

Molecular Formula C20H19ClN6O3
MW 426.86
Aromatic Rings 4
Heavy Atoms 30
NP-Likeness -1.35

Activity Summary

IC50 4 meas. best 8.41

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Transient receptor potential cation channel subfamily A member 1
CHEMBL6007
IC50 8.41 8.215 3.9 4

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine