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Compound Detail

CHEMBL5946660

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CCC1(CC)C=Cc2c(ccc(C=O)c2OC(=O)c2ccccc2)O1

Basic Information

ChEMBL ID CHEMBL5946660
Phase Preclinical
Structure Type MOL
InChI Key DOSGAQQUQFVYLL-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

336.4
MW (Da)
4.68
ALogP
4
HBA
0
HBD
52.6
PSA (Ų)
0.45
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H20O4
MW 336.39
Aromatic Rings 2
Heavy Atoms 25
NP-Likeness 0.95

Activity Summary

IC50 1 meas. best 5.19

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Tyrosine-protein phosphatase non-receptor type 1
CHEMBL335
IC50 5.19 5.19 6500.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine