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Compound Detail

CHEMBL5990651

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CN(C)c1ccc(C#Cc2cc3cc(F)cnc3[nH]2)cc1

Basic Information

ChEMBL ID CHEMBL5990651
Phase Preclinical
Structure Type MOL
InChI Key XJKFPLBHLHQERY-UHFFFAOYSA-N
2
Targets
2
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

279.3
MW (Da)
3.17
ALogP
2
HBA
1
HBD
31.9
PSA (Ų)
0.69
QED
0
Ro5 Violations
1
Rot. Bonds

Drug Information

Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C17H14FN3
MW 279.32
Aromatic Rings 3
Heavy Atoms 21
NP-Likeness -1.19

Activity Summary

Ki 2 meas. best 7.72

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Alpha-synuclein
CHEMBL6152
Ki 7.72 7.72 19.0 1
Unchecked
CHEMBL612545
Ki 6.5 6.5 318.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine