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Compound Detail

CHEMBL609180

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OC1O[C@H](CSc2ccc(F)cc2)[C@@H](O)[C@H]1O

Basic Information

ChEMBL ID CHEMBL609180
Phase Preclinical
Structure Type MOL
InChI Key PJYDYUDAULCICX-QHPFDFDXSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
10
Publications
0
Known Names

Molecular Properties

260.3
MW (Da)
0.36
ALogP
5
HBA
3
HBD
69.9
PSA (Ų)
0.68
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C11H13FO4S
MW 260.29
Aromatic Rings 1
Heavy Atoms 17
NP-Likeness 0.31

Activity Summary

IC50 1 meas. best 10.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Klebsiella pneumoniae
CHEMBL350
IC50 10.3 10.3 0.1 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Klebsiella pneumoniae IC50 = 0.05 nM 10.3 Compound was tested for its ability to inhibit the growth of a clinical strain o... -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(01)81020-9 Klebsiella pneumoniae 2
- 10.6019/CHEMBL4513161 Pseudomonas aeruginosa 2
- 10.6019/CHEMBL4513161 Candida albicans 1
- 10.6019/CHEMBL4513161 Cryptococcus neoformans 1
- 10.6019/CHEMBL4513161 Escherichia coli 1
- 10.6019/CHEMBL4513161 Klebsiella pneumoniae 1
- 10.6019/CHEMBL4513161 Acinetobacter baumannii 1
- 10.6019/CHEMBL4513161 Staphylococcus aureus 1
- 10.6019/CHEMBL4513161 Erythrocyte 1
- 10.6019/CHEMBL4513161 HEK293 1

Data from ChEMBL 36 via Core Engine