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Compound Detail

CHEMBL7026

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O=C1OC(=O)[C@@H]2[C@H]1[C@@H]1O[C@H]2C[C@@H]1COC(=O)[C@@H]1C[C@H]1c1ccccc1

Basic Information

ChEMBL ID CHEMBL7026
Phase Preclinical
Structure Type MOL
InChI Key OFHGSESHXNRPRM-NMCQGECBSA-N
1
Targets
2
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

342.4
MW (Da)
1.44
ALogP
6
HBA
0
HBD
78.9
PSA (Ų)
0.61
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C19H18O6
MW 342.35
Aromatic Rings 1
Heavy Atoms 25
NP-Likeness 0.67

Activity Summary

Ki 2 meas. best 6.3

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
Ki 6.3 5.85 500.0 2

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked Ki = 500.0 nM 6.3 Inhibition of Protein phosphatase 2B -
Unchecked Ki = 4000.0 nM 5.4 The compound was tested for the inhibition of Protein phosphatase-1 (PP1) -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(97)00141-8 Unchecked 2

Data from ChEMBL 36 via Core Engine