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Compound Detail

CHEMBL96189

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O=C(NC[C@H](NS(=O)(=O)c1cccnc1)C(=O)O)c1cc2c(s1)CCN(CCC1CCNCC1)C2=O

Basic Information

ChEMBL ID CHEMBL96189
Phase Preclinical
Structure Type MOL
InChI Key XJDGTXWATZIYJY-SFHVURJKSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

535.6
MW (Da)
0.69
ALogP
8
HBA
4
HBD
157.8
PSA (Ų)
0.35
QED
1
Ro5 Violations
10
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C23H29N5O6S2
MW 535.65
Aromatic Rings 2
Heavy Atoms 36
NP-Likeness -1.26

Activity Summary

IC50 1 meas. best 7.89

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Homo sapiens
CHEMBL372
IC50 7.89 7.89 13.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Homo sapiens IC50 = 13.0 nM 7.89 Compound was evaluated for inhibition of ex vivo ADP mediated platelet aggregati... -

Literature References

PubMed DOI Target Context # Activities
- 10.1016/S0960-894X(96)00511-2 Homo sapiens 1

Data from ChEMBL 36 via Core Engine