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Compound Detail

CHEMBL9807

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COP(=O)(Nc1ccc(Nc2c3ccccc3nc3ccccc23)cc1)OC

Basic Information

ChEMBL ID CHEMBL9807
Phase Preclinical
Structure Type MOL
InChI Key ZBXGOHXTOZVTDQ-UHFFFAOYSA-N
1
Targets
1
Activities
1
Assay Types
0
PK Parameters
8
Publications
0
Known Names

Molecular Properties

393.4
MW (Da)
5.94
ALogP
5
HBA
2
HBD
72.5
PSA (Ų)
0.31
QED
1
Ro5 Violations
6
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H20N3O3P
MW 393.38
Aromatic Rings 4
Heavy Atoms 28
NP-Likeness -0.43

Activity Summary

IC50 1 meas. best 7.82

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
L1210
CHEMBL386
IC50 7.82 7.82 15.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
L1210 IC50 = 15.0 nM 7.82 Inhibitory concentration to reduce the growth of L1210 cells by 50% after 70 hr.... 3820217

Literature References

Data from ChEMBL 36 via Core Engine