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Assay Detail

CHEMBL1002235

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of human recombinant CYP2C9 expressed in insect microsomes
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Subcellular Microsome
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 2C9 (CHEMBL3397)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Overcoming undesirable CYP1A2 inhibition of pyridylnaphthalene-type aldosterone synthase inhibitors: influence of heteroaryl derivatization on potency and selectivity.
Heim R, Lucas S, Grombein CM, Ries C, Schewe KE, Negri M, Müller-Vieira U, Birk B, Hartmann RW.
J Med Chem (2008) 51 : 5064 -5074
PubMed 18672861 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.61 6.50

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1109 SULFAPHENAZOLE 4.0 1 6.50
CHEMBL500394 1 5.90
CHEMBL447591 1 5.72
CHEMBL453169 1 4.31
CHEMBL502824 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1109 SULFAPHENAZOLE IC50 = 318.0 nM 6.50
CHEMBL500394 IC50 = 1270.0 nM 5.90
CHEMBL447591 IC50 = 1888.0 nM 5.72
CHEMBL453169 IC50 = 48970.0 nM 4.31
CHEMBL502824 IC50 > 200000.0 nM -