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Assay Detail

CHEMBL1020883

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Binding
Inhibition of 5HT uptake at rat brain SERT
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Rattus norvegicus
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sodium-dependent serotonin transporter (CHEMBL313)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Structure-activity relationships of the cycloalkanol ethylamine scaffold: discovery of selective norepinephrine reuptake inhibitors.
Mahaney PE, Gavrin LK, Trybulski EJ, Stack GP, Vu TA, Cohn ST, Ye F, Belardi JK, Santilli AA, Sabatucci JP, Leiter J, Johnston GH, Bray JA, Burroughs KD, Cosmi SA, Leventhal L, Koury EJ, Zhang Y, Mugford CA, Ho DM, Rosenzweig-Lipson SJ, Platt B, Smith VA, Deecher DC.
J Med Chem (2008) 51 : 4038 -4049
PubMed 18557608 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 6.73 7.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL316862 1 7.89
CHEMBL420644 1 6.75
CHEMBL101055 1 6.72
CHEMBL637 VENLAFAXINE 4.0 1 6.68
CHEMBL101899 1 6.50
CHEMBL99653 1 5.84

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL316862 IC50 = 13.0 nM 7.89
CHEMBL420644 IC50 = 180.0 nM 6.75
CHEMBL101055 IC50 = 190.0 nM 6.72
CHEMBL637 VENLAFAXINE IC50 = 210.0 nM 6.68
CHEMBL101899 IC50 = 320.0 nM 6.50
CHEMBL99653 IC50 = 1440.0 nM 5.84