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Assay Detail

CHEMBL1101481

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of serotonin uptake at human SERT expressed in human JAR
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sodium-dependent serotonin transporter (CHEMBL228)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structure-activity relationships of norepinephrine reuptake inhibitors with benzothiadiazine dioxide or dihydrosulfostyril cores.
Fensome A, Goldberg J, McComas CC, Trybulski EJ, Woodworth RP, Deecher DC, Whiteside GT, Zhang P.
Bioorg Med Chem Lett (2010) 20 : 1555 -1558
PubMed 20153188 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 13 5.78 6.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1083211 1 6.96
CHEMBL1204413 1 6.62
CHEMBL1204414 1 6.47
CHEMBL1204415 1 6.22
CHEMBL1096001 1 6.14
CHEMBL1083210 1 5.82
CHEMBL1084933 1 5.70
CHEMBL1204410 1 5.60
CHEMBL1087924 1 5.26
CHEMBL1086398 1 5.22
CHEMBL1077209 1 5.16
CHEMBL1204412 1 5.10
CHEMBL1084934 1 4.88

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1083211 IC50 = 110.0 nM 6.96
CHEMBL1204413 IC50 = 240.0 nM 6.62
CHEMBL1204414 IC50 = 340.0 nM 6.47
CHEMBL1204415 IC50 = 600.0 nM 6.22
CHEMBL1096001 IC50 = 720.0 nM 6.14
CHEMBL1083210 IC50 = 1500.0 nM 5.82
CHEMBL1084933 IC50 = 2000.0 nM 5.70
CHEMBL1204410 IC50 = 2500.0 nM 5.60
CHEMBL1087924 IC50 = 5500.0 nM 5.26
CHEMBL1086398 IC50 = 6000.0 nM 5.22
CHEMBL1077209 IC50 = 6900.0 nM 5.16
CHEMBL1204412 IC50 = 8000.0 nM 5.10
CHEMBL1084934 IC50 = 13300.0 nM 4.88