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Assay Detail

CHEMBL1106978

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]N-methylscopolamine from human muscarinic M1 receptor expressed in CHO Flp-In cells after 90 mins by scintillation counting
29
Total Activities
29
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Muscarinic acetylcholine receptor M1 (CHEMBL216)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Novel benzothiophene H1-antihistamines for the treatment of insomnia.
Moree WJ, Jovic F, Coon T, Yu J, Li BF, Tucci FC, Marinkovic D, Gross RS, Malany S, Bradbury MJ, Hernandez LM, O'Brien Z, Wen J, Wang H, Hoare SR, Petroski RE, Sacaan A, Madan A, Crowe PD, Beaton G.
Bioorg Med Chem Lett (2010) 20 : 2316 -2320
PubMed 20188547 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 25 6.43 8.25
IC50 4 5.35 5.43

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1091790 1 8.25
CHEMBL1091774 1 8.24
CHEMBL1090433 1 6.00
CHEMBL1090432 1 5.85
CHEMBL1092377 1 5.66
CHEMBL1093044 1 5.43
CHEMBL1091776 1 5.33
CHEMBL564144 1 5.28
CHEMBL1091777 1 4.55
CHEMBL1092496 1 -
CHEMBL1092495 1 -
CHEMBL1092494 1 -
CHEMBL1091069 1 -
CHEMBL1092126 1 -
CHEMBL1091793 1 -
CHEMBL1091792 1 -
CHEMBL1091791 1 -
CHEMBL1091778 1 -
CHEMBL1091775 1 -
CHEMBL1092812 1 -
CHEMBL1092813 1 -
CHEMBL1093294 1 -
CHEMBL1093058 1 -
CHEMBL1092765 1 -
CHEMBL1092766 1 -
CHEMBL1092767 1 -
CHEMBL1091782 1 -
CHEMBL1092118 1 -
CHEMBL1093607 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1091790 Ki = 5.6 nM 8.25
CHEMBL1091774 Ki = 5.8 nM 8.24
CHEMBL1090433 Ki = 990.0 nM 6.00
CHEMBL1090432 Ki = 1400.0 nM 5.85
CHEMBL1092377 Ki = 2200.0 nM 5.66
CHEMBL1093044 IC50 = 3700.0 nM 5.43
CHEMBL1091776 IC50 = 4700.0 nM 5.33
CHEMBL564144 IC50 = 5300.0 nM 5.28
CHEMBL1091777 Ki = 28000.0 nM 4.55
CHEMBL1092496 Ki > 10000.0 nM -
CHEMBL1092495 Ki > 10000.0 nM -
CHEMBL1092494 Ki > 10000.0 nM -
CHEMBL1091069 Ki > 10000.0 nM -
CHEMBL1092126 Ki > 10000.0 nM -
CHEMBL1091793 Ki > 10000.0 nM -
CHEMBL1091792 Ki > 10000.0 nM -
CHEMBL1091791 Ki > 10000.0 nM -
CHEMBL1091778 IC50 > 10000.0 nM -
CHEMBL1091775 Ki > 10000.0 nM -
CHEMBL1092812 Ki > 10000.0 nM -
CHEMBL1092813 Ki > 10000.0 nM -
CHEMBL1093294 Ki > 10000.0 nM -
CHEMBL1093058 Ki > 10000000.0 nM -
CHEMBL1092765 Ki > 10000.0 nM -
CHEMBL1092766 Ki > 10000.0 nM -
CHEMBL1092767 Ki = 2072000.0 nM -
CHEMBL1091782 Ki = 4759000.0 nM -
CHEMBL1092118 Ki > 10000000.0 nM -
CHEMBL1093607 Ki - -