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Assay Detail

CHEMBL1110024

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]citalopram form human SRET by liquid scintillation counting
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Sodium-dependent serotonin transporter (CHEMBL228)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Potent dihydroquinolinone dopamine D2 partial agonist/serotonin reuptake inhibitors for the treatment of schizophrenia.
Yan Y, Zhou P, Rotella DP, Feenstra R, Kruse CG, Reinders JH, van der Neut M, Lai M, Zhang J, Kowal DM, Carrick T, Marquis KL, Pausch MH, Robichaud AJ.
Bioorg Med Chem Lett (2010) 20 : 2983 -2986
PubMed 20347298 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 14 7.99 9.59

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1088000 1 9.59
CHEMBL1508 ESCITALOPRAM 4.0 1 9.00
CHEMBL1087817 1 8.82
CHEMBL1087818 1 8.77
CHEMBL1087455 1 8.72
CHEMBL1087585 1 8.30
CHEMBL1088560 1 7.72
CHEMBL1087744 1 7.70
CHEMBL1087743 1 7.70
CHEMBL1087745 1 7.66
CHEMBL1087872 1 7.52
CHEMBL1087454 1 7.03
CHEMBL1087453 1 7.03
CHEMBL1087452 1 6.27

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1088000 Ki = 0.26 nM 9.59
CHEMBL1508 ESCITALOPRAM Ki = 1.0 nM 9.00
CHEMBL1087817 Ki = 1.5 nM 8.82
CHEMBL1087818 Ki = 1.7 nM 8.77
CHEMBL1087455 Ki = 1.9 nM 8.72
CHEMBL1087585 Ki = 5.0 nM 8.30
CHEMBL1088560 Ki = 19.0 nM 7.72
CHEMBL1087744 Ki = 20.0 nM 7.70
CHEMBL1087743 Ki = 20.0 nM 7.70
CHEMBL1087745 Ki = 22.0 nM 7.66
CHEMBL1087872 Ki = 30.0 nM 7.52
CHEMBL1087454 Ki = 94.0 nM 7.03
CHEMBL1087453 Ki = 93.0 nM 7.03
CHEMBL1087452 Ki = 538.0 nM 6.27