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Assay Detail

CHEMBL1284240

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against herpes simplex virus 1 E-377 infected in HFF cells by plaque reduction assay
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 1
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Target

Human alphaherpesvirus 1 (CHEMBL377)
Type ORGANISM
Organism Human alphaherpesvirus 1

Publication

Inhibition of herpesvirus replication by hexadecyloxypropyl esters of purine- and pyrimidine-based phosphonomethoxyethyl nucleoside phosphonates.
Prichard MN, Hartline CB, Harden EA, Daily SL, Beadle JR, Valiaeva N, Kern ER, Hostetler KY.
Antimicrob Agents Chemother (2008) 52 : 4326 -4330
PubMed 18852272 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 10 6.14 7.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL502317 1 7.00
CHEMBL473586 1 6.22
CHEMBL1276695 1 5.92
CHEMBL223160 1 5.40
CHEMBL1275686 1 -
CHEMBL63849 1 -
CHEMBL418216 1 -
CHEMBL1276696 1 -
CHEMBL61733 PMEDAP 1 -
CHEMBL1276665 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL502317 EC50 = 100.0 nM 7.00
CHEMBL473586 EC50 = 600.0 nM 6.22
CHEMBL1276695 EC50 = 1200.0 nM 5.92
CHEMBL223160 EC50 = 4000.0 nM 5.40
CHEMBL1275686 EC50 - -
CHEMBL63849 EC50 > 60000.0 nM -
CHEMBL418216 EC50 > 300000.0 nM -
CHEMBL1276696 EC50 > 12000.0 nM -
CHEMBL61733 PMEDAP EC50 > 10000.0 nM -
CHEMBL1276665 EC50 = 260000.0 nM -