Assay Detail
Functional
CHEMBL1613839
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response HTS to Identify Activators of Luciferase Translation or Activity in H4-C Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1829 (Project Summary), 1814 (Primary HTS)]
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 40 | 5.69 | 6.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1410134 | — | — | 1 | 6.68 |
| CHEMBL1331904 | — | — | 1 | 6.61 |
| CHEMBL1331733 | — | — | 1 | 6.25 |
| CHEMBL1377188 | — | — | 1 | 6.21 |
| CHEMBL1408486 | — | — | 1 | 6.20 |
| CHEMBL1522289 | — | — | 1 | 6.16 |
| CHEMBL1371056 | — | — | 1 | 6.15 |
| CHEMBL1476311 | — | — | 1 | 6.11 |
| CHEMBL1354093 | — | — | 1 | 6.04 |
| CHEMBL1316021 | — | — | 1 | 6.03 |
| CHEMBL1493731 | — | — | 1 | 6.02 |
| CHEMBL1476264 | — | — | 1 | 5.98 |
| CHEMBL1369984 | — | — | 1 | 5.98 |
| CHEMBL1330793 | — | — | 1 | 5.97 |
| CHEMBL1513325 | — | — | 1 | 5.94 |
| CHEMBL1300558 | — | — | 1 | 5.87 |
| CHEMBL1389580 | — | — | 1 | 5.83 |
| CHEMBL1488300 | — | — | 1 | 5.79 |
| CHEMBL1407944 | — | — | 1 | 5.76 |
| CHEMBL1452245 | — | — | 1 | 5.73 |
| CHEMBL1448972 | — | — | 1 | 5.68 |
| CHEMBL1313968 | — | — | 1 | 5.67 |
| CHEMBL1409108 | — | — | 1 | 5.67 |
| CHEMBL1620207 | — | — | 1 | 5.67 |
| CHEMBL1391573 | — | — | 1 | 5.63 |
| CHEMBL602722 | — | — | 1 | 5.63 |
| CHEMBL1358278 | — | — | 1 | 5.60 |
| CHEMBL1314043 | — | — | 1 | 5.57 |
| CHEMBL1569667 | — | — | 1 | 5.54 |
| CHEMBL1331836 | — | — | 1 | 5.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1410134 | — | EC50 | = | 207.0 | nM | 6.68 |
| CHEMBL1331904 | — | EC50 | = | 246.0 | nM | 6.61 |
| CHEMBL1331733 | — | EC50 | = | 557.0 | nM | 6.25 |
| CHEMBL1377188 | — | EC50 | = | 609.0 | nM | 6.21 |
| CHEMBL1408486 | — | EC50 | = | 630.0 | nM | 6.20 |
| CHEMBL1522289 | — | EC50 | = | 697.0 | nM | 6.16 |
| CHEMBL1371056 | — | EC50 | = | 703.0 | nM | 6.15 |
| CHEMBL1476311 | — | EC50 | = | 772.0 | nM | 6.11 |
| CHEMBL1354093 | — | EC50 | = | 921.0 | nM | 6.04 |
| CHEMBL1316021 | — | EC50 | = | 929.0 | nM | 6.03 |
| CHEMBL1493731 | — | EC50 | = | 946.0 | nM | 6.02 |
| CHEMBL1476264 | — | EC50 | = | 1049.0 | nM | 5.98 |
| CHEMBL1369984 | — | EC50 | = | 1056.0 | nM | 5.98 |
| CHEMBL1330793 | — | EC50 | = | 1074.0 | nM | 5.97 |
| CHEMBL1513325 | — | EC50 | = | 1156.0 | nM | 5.94 |
| CHEMBL1300558 | — | EC50 | = | 1365.0 | nM | 5.87 |
| CHEMBL1389580 | — | EC50 | = | 1464.0 | nM | 5.83 |
| CHEMBL1488300 | — | EC50 | = | 1630.0 | nM | 5.79 |
| CHEMBL1407944 | — | EC50 | = | 1745.0 | nM | 5.76 |
| CHEMBL1452245 | — | EC50 | = | 1880.0 | nM | 5.73 |
| CHEMBL1448972 | — | EC50 | = | 2065.0 | nM | 5.68 |
| CHEMBL1409108 | — | EC50 | = | 2146.0 | nM | 5.67 |
| CHEMBL1620207 | — | EC50 | = | 2123.0 | nM | 5.67 |
| CHEMBL1313968 | — | EC50 | = | 2139.0 | nM | 5.67 |
| CHEMBL1391573 | — | EC50 | = | 2330.0 | nM | 5.63 |
| CHEMBL602722 | — | EC50 | = | 2323.0 | nM | 5.63 |
| CHEMBL1358278 | — | EC50 | = | 2510.0 | nM | 5.60 |
| CHEMBL1314043 | — | EC50 | = | 2691.0 | nM | 5.57 |
| CHEMBL1569667 | — | EC50 | = | 2906.0 | nM | 5.54 |
| CHEMBL1376513 | — | EC50 | = | 2956.0 | nM | 5.53 |
| CHEMBL1331836 | — | EC50 | = | 2966.0 | nM | 5.53 |
| CHEMBL1329938 | — | EC50 | = | 3069.0 | nM | 5.51 |
| CHEMBL1440659 | — | EC50 | = | 4388.0 | nM | 5.36 |
| CHEMBL1528120 | — | EC50 | = | 6810.0 | nM | 5.17 |
| CHEMBL1354131 | — | EC50 | = | 10282.0 | nM | 4.99 |
| CHEMBL1414223 | — | EC50 | = | 13210.0 | nM | 4.88 |
| CHEMBL1490480 | — | EC50 | = | 20469.0 | nM | 4.69 |
| CHEMBL1349455 | — | EC50 | = | 51134.0 | nM | 4.29 |
| CHEMBL1555236 | — | EC50 | = | 73124.0 | nM | 4.14 |
| CHEMBL1304057 | — | EC50 | > | 195000.0 | nM | - |