Assay Detail
Binding
CHEMBL1613844
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of PP5: fluorescence-based biochemical high throughput dose response assay for inhibitors of Protein Phosphatase 1 (PP1). (Class of assay: confirmatory) [Related pubchem assays: 2034 (Summary (PP5 inhibitors)), 1987 (Primary screen (PP5 inhibitors)), 2235 (Screening assay (PP1 inhibitors in singlate))]
60
Total Activities
60
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Serine/threonine-protein phosphatase PP1-alpha catalytic subunit (CHEMBL2164) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 60 | 4.46 | 5.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL567967 | — | — | 1 | 5.57 |
| CHEMBL2003651 | — | — | 1 | 4.81 |
| CHEMBL2003806 | — | — | 1 | 4.73 |
| CHEMBL1898479 | — | — | 1 | 4.67 |
| CHEMBL3190880 | — | — | 1 | 4.64 |
| CHEMBL1969046 | — | — | 1 | 4.57 |
| CHEMBL1412774 | — | — | 1 | 4.55 |
| CHEMBL3144999 | — | — | 1 | 4.52 |
| CHEMBL1299200 | — | — | 1 | 4.49 |
| CHEMBL3196591 | — | — | 1 | 4.46 |
| CHEMBL175434 | — | — | 1 | 4.41 |
| CHEMBL2006503 | — | — | 1 | 4.41 |
| CHEMBL1426692 | — | — | 1 | 4.36 |
| CHEMBL1530147 | — | — | 1 | 4.36 |
| CHEMBL1453503 | — | — | 1 | 4.33 |
| CHEMBL1410383 | — | — | 1 | 4.33 |
| CHEMBL1577193 | — | — | 1 | 4.31 |
| CHEMBL1501990 | — | — | 1 | 4.31 |
| CHEMBL1598762 | — | — | 1 | 4.28 |
| CHEMBL1397706 | — | — | 1 | 4.28 |
| CHEMBL1536273 | — | — | 1 | 4.25 |
| CHEMBL1450505 | — | — | 1 | 4.24 |
| CHEMBL1362561 | — | — | 1 | 4.20 |
| CHEMBL1463829 | — | — | 1 | 4.20 |
| CHEMBL1477061 | — | — | 1 | 4.19 |
| CHEMBL1902079 | — | — | 1 | - |
| CHEMBL1996724 | — | — | 1 | - |
| CHEMBL1562466 | — | — | 1 | - |
| CHEMBL1378634 | — | — | 1 | - |
| CHEMBL3194941 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL567967 | — | IC50 | = | 2667.0 | nM | 5.57 |
| CHEMBL2003651 | — | IC50 | = | 15546.0 | nM | 4.81 |
| CHEMBL2003806 | — | IC50 | = | 18550.0 | nM | 4.73 |
| CHEMBL1898479 | — | IC50 | = | 21556.0 | nM | 4.67 |
| CHEMBL3190880 | — | IC50 | = | 22658.0 | nM | 4.64 |
| CHEMBL1969046 | — | IC50 | = | 27075.0 | nM | 4.57 |
| CHEMBL1412774 | — | IC50 | = | 28288.0 | nM | 4.55 |
| CHEMBL3144999 | — | IC50 | = | 29894.0 | nM | 4.52 |
| CHEMBL1299200 | — | IC50 | = | 32124.0 | nM | 4.49 |
| CHEMBL3196591 | — | IC50 | = | 34360.0 | nM | 4.46 |
| CHEMBL175434 | — | IC50 | = | 38859.0 | nM | 4.41 |
| CHEMBL2006503 | — | IC50 | = | 38913.0 | nM | 4.41 |
| CHEMBL1426692 | — | IC50 | = | 44079.0 | nM | 4.36 |
| CHEMBL1530147 | — | IC50 | = | 43617.0 | nM | 4.36 |
| CHEMBL1410383 | — | IC50 | = | 46188.0 | nM | 4.33 |
| CHEMBL1453503 | — | IC50 | = | 46923.0 | nM | 4.33 |
| CHEMBL1577193 | — | IC50 | = | 49020.0 | nM | 4.31 |
| CHEMBL1501990 | — | IC50 | = | 48978.0 | nM | 4.31 |
| CHEMBL1598762 | — | IC50 | = | 52139.0 | nM | 4.28 |
| CHEMBL1397706 | — | IC50 | = | 52346.0 | nM | 4.28 |
| CHEMBL1536273 | — | IC50 | = | 56486.0 | nM | 4.25 |
| CHEMBL1450505 | — | IC50 | = | 57600.0 | nM | 4.24 |
| CHEMBL1362561 | — | IC50 | = | 63577.0 | nM | 4.20 |
| CHEMBL1463829 | — | IC50 | = | 62464.0 | nM | 4.20 |
| CHEMBL1477061 | — | IC50 | = | 64048.0 | nM | 4.19 |
| CHEMBL1432243 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL205040 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1392911 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1432553 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1495013 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1502394 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1303854 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1402456 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1334040 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1361173 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1346300 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL3189714 | — | IC50 | > | 22349.0 | nM | - |
| CHEMBL1516601 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1563939 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL578905 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1446100 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1379448 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1585740 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1516738 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1458321 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL3194941 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1378634 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1562466 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1996724 | — | IC50 | > | 67047.0 | nM | - |
| CHEMBL1902079 | — | IC50 | > | 67047.0 | nM | - |