Assay Detail
Functional
CHEMBL1613871
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response to Identify Inhibitors of Luciferase Translation or Activity in H4-C Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1813 (Primary HTS), 1827 (Project Summary)]
183
Total Activities
183
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 183 | 6.47 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1555935 | — | — | 1 | 8.30 |
| CHEMBL3192138 | — | — | 1 | 8.10 |
| CHEMBL1462938 | — | — | 1 | 8.05 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 7.82 |
| CHEMBL1562575 | — | — | 1 | 7.82 |
| CHEMBL1536981 | — | — | 1 | 7.68 |
| CHEMBL513000 | — | — | 1 | 7.52 |
| CHEMBL1342336 | — | — | 1 | 7.47 |
| CHEMBL1751 | DIGOXIN | 4.0 | 1 | 7.47 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.41 |
| CHEMBL1307091 | — | — | 1 | 7.36 |
| CHEMBL501867 | VINCRISTINE SULFATE | 4.0 | 1 | 7.33 |
| CHEMBL1495092 | — | — | 1 | 7.30 |
| CHEMBL1537509 | — | — | 1 | 7.29 |
| CHEMBL1368103 | — | — | 1 | 7.29 |
| CHEMBL1347346 | — | — | 1 | 7.24 |
| CHEMBL3185655 | — | — | 1 | 7.23 |
| CHEMBL1357620 | — | — | 1 | 7.21 |
| CHEMBL1521023 | — | — | 1 | 7.17 |
| CHEMBL1587117 | — | — | 1 | 7.14 |
| CHEMBL300389 | — | — | 1 | 7.13 |
| CHEMBL1376974 | — | — | 1 | 7.13 |
| CHEMBL1987060 | — | — | 1 | 7.11 |
| CHEMBL312862 | DEMECOLCINE | 2.0 | 1 | 7.11 |
| CHEMBL222863 | OUABAIN | -1.0 | 1 | 7.08 |
| CHEMBL1355541 | — | — | 1 | 7.08 |
| CHEMBL1884996 | — | — | 1 | 7.08 |
| CHEMBL3195389 | — | — | 1 | 7.07 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | -1.0 | 1 | 7.06 |
| CHEMBL1595169 | — | — | 1 | 7.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1555935 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL3192138 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL1462938 | — | EC50 | = | 9.0 | nM | 8.05 |
| CHEMBL1562575 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL61 | PODOFILOX | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL1536981 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL513000 | — | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL1751 | DIGOXIN | EC50 | = | 34.0 | nM | 7.47 |
| CHEMBL1342336 | — | EC50 | = | 34.0 | nM | 7.47 |
| CHEMBL428647 | PACLITAXEL | EC50 | = | 39.0 | nM | 7.41 |
| CHEMBL1307091 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL501867 | VINCRISTINE SULFATE | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL1495092 | — | EC50 | = | 50.0 | nM | 7.30 |
| CHEMBL1368103 | — | EC50 | = | 51.0 | nM | 7.29 |
| CHEMBL1537509 | — | EC50 | = | 51.0 | nM | 7.29 |
| CHEMBL1347346 | — | EC50 | = | 58.0 | nM | 7.24 |
| CHEMBL3185655 | — | EC50 | = | 59.0 | nM | 7.23 |
| CHEMBL1357620 | — | EC50 | = | 62.0 | nM | 7.21 |
| CHEMBL1521023 | — | EC50 | = | 67.0 | nM | 7.17 |
| CHEMBL1587117 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1376974 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL300389 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL312862 | DEMECOLCINE | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1987060 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1884996 | — | EC50 | = | 84.0 | nM | 7.08 |
| CHEMBL222863 | OUABAIN | EC50 | = | 84.0 | nM | 7.08 |
| CHEMBL1355541 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL3195389 | — | EC50 | = | 86.0 | nM | 7.07 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | EC50 | = | 88.0 | nM | 7.06 |
| CHEMBL1595169 | — | EC50 | = | 87.0 | nM | 7.06 |
| CHEMBL423192 | ANISOMYCIN | EC50 | = | 91.0 | nM | 7.04 |
| CHEMBL1473676 | — | EC50 | = | 92.0 | nM | 7.04 |
| CHEMBL373137 | — | EC50 | = | 96.0 | nM | 7.02 |
| CHEMBL1333930 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1392142 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL460601 | — | EC50 | = | 103.0 | nM | 6.99 |
| CHEMBL1537098 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1256472 | CYTARABINE HYDROCHLORIDE | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1323774 | — | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL1602385 | — | EC50 | = | 111.0 | nM | 6.96 |
| CHEMBL1405749 | — | EC50 | = | 113.0 | nM | 6.95 |
| CHEMBL1372889 | — | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL579318 | — | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL1423192 | — | EC50 | = | 126.0 | nM | 6.90 |
| CHEMBL1528660 | — | EC50 | = | 125.0 | nM | 6.90 |
| CHEMBL1453996 | — | EC50 | = | 134.0 | nM | 6.87 |
| CHEMBL1312738 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL1483593 | — | EC50 | = | 143.0 | nM | 6.84 |
| CHEMBL1316831 | — | EC50 | = | 157.0 | nM | 6.80 |
| CHEMBL9514 | NOCODAZOLE | EC50 | = | 195.0 | nM | 6.71 |