Assay Detail
Functional
CHEMBL1613878
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Retest to Confirm Activators of 5'UTR Stem-Loop Driven Alpha-Synuclein mRNA Translation in H4 Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1813, AID1829]
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 38 | 5.39 | 6.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1522289 | — | — | 1 | 6.18 |
| CHEMBL1476264 | — | — | 1 | 6.17 |
| CHEMBL1376513 | — | — | 1 | 6.14 |
| CHEMBL1488300 | — | — | 1 | 6.12 |
| CHEMBL1389580 | — | — | 1 | 6.09 |
| CHEMBL1452245 | — | — | 1 | 6.05 |
| CHEMBL1448972 | — | — | 1 | 6.04 |
| CHEMBL1409108 | — | — | 1 | 5.88 |
| CHEMBL1331733 | — | — | 1 | 5.78 |
| CHEMBL1316021 | — | — | 1 | 5.75 |
| CHEMBL602722 | — | — | 1 | 5.75 |
| CHEMBL1412667 | — | — | 1 | 5.74 |
| CHEMBL1354093 | — | — | 1 | 5.73 |
| CHEMBL1620207 | — | — | 1 | 5.73 |
| CHEMBL1329938 | — | — | 1 | 5.73 |
| CHEMBL1369984 | — | — | 1 | 5.69 |
| CHEMBL1407944 | — | — | 1 | 5.68 |
| CHEMBL1513325 | — | — | 1 | 5.57 |
| CHEMBL1391573 | — | — | 1 | 5.54 |
| CHEMBL1313968 | — | — | 1 | 5.21 |
| CHEMBL1354131 | — | — | 1 | 5.20 |
| CHEMBL1330793 | — | — | 1 | 5.13 |
| CHEMBL1331904 | — | — | 1 | 5.03 |
| CHEMBL1569667 | — | — | 1 | 4.93 |
| CHEMBL1490480 | — | — | 1 | 4.78 |
| CHEMBL1440659 | — | — | 1 | 4.67 |
| CHEMBL1493731 | — | — | 1 | 4.65 |
| CHEMBL1314043 | — | — | 1 | 4.58 |
| CHEMBL1300558 | — | — | 1 | 4.58 |
| CHEMBL1358278 | — | — | 1 | 4.53 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1522289 | — | EC50 | = | 666.0 | nM | 6.18 |
| CHEMBL1476264 | — | EC50 | = | 673.0 | nM | 6.17 |
| CHEMBL1376513 | — | EC50 | = | 719.0 | nM | 6.14 |
| CHEMBL1488300 | — | EC50 | = | 752.0 | nM | 6.12 |
| CHEMBL1389580 | — | EC50 | = | 811.0 | nM | 6.09 |
| CHEMBL1452245 | — | EC50 | = | 885.0 | nM | 6.05 |
| CHEMBL1448972 | — | EC50 | = | 901.0 | nM | 6.04 |
| CHEMBL1409108 | — | EC50 | = | 1314.0 | nM | 5.88 |
| CHEMBL1331733 | — | EC50 | = | 1661.0 | nM | 5.78 |
| CHEMBL1316021 | — | EC50 | = | 1775.0 | nM | 5.75 |
| CHEMBL602722 | — | EC50 | = | 1760.0 | nM | 5.75 |
| CHEMBL1412667 | — | EC50 | = | 1807.0 | nM | 5.74 |
| CHEMBL1354093 | — | EC50 | = | 1844.0 | nM | 5.73 |
| CHEMBL1620207 | — | EC50 | = | 1877.0 | nM | 5.73 |
| CHEMBL1329938 | — | EC50 | = | 1849.0 | nM | 5.73 |
| CHEMBL1369984 | — | EC50 | = | 2036.0 | nM | 5.69 |
| CHEMBL1407944 | — | EC50 | = | 2089.0 | nM | 5.68 |
| CHEMBL1513325 | — | EC50 | = | 2694.0 | nM | 5.57 |
| CHEMBL1391573 | — | EC50 | = | 2861.0 | nM | 5.54 |
| CHEMBL1313968 | — | EC50 | = | 6154.0 | nM | 5.21 |
| CHEMBL1354131 | — | EC50 | = | 6356.0 | nM | 5.20 |
| CHEMBL1330793 | — | EC50 | = | 7373.0 | nM | 5.13 |
| CHEMBL1331904 | — | EC50 | = | 9275.0 | nM | 5.03 |
| CHEMBL1569667 | — | EC50 | = | 11632.0 | nM | 4.93 |
| CHEMBL1490480 | — | EC50 | = | 16551.0 | nM | 4.78 |
| CHEMBL1440659 | — | EC50 | = | 21480.0 | nM | 4.67 |
| CHEMBL1493731 | — | EC50 | = | 22543.0 | nM | 4.65 |
| CHEMBL1314043 | — | EC50 | = | 26331.0 | nM | 4.58 |
| CHEMBL1300558 | — | EC50 | = | 26600.0 | nM | 4.58 |
| CHEMBL1358278 | — | EC50 | = | 29524.0 | nM | 4.53 |
| CHEMBL1528120 | — | EC50 | = | 33359.0 | nM | 4.48 |
| CHEMBL1331836 | — | EC50 | = | 35780.0 | nM | 4.45 |
| CHEMBL1371056 | — | EC50 | = | 36363.0 | nM | 4.44 |
| CHEMBL1414223 | — | EC50 | > | 195000.0 | nM | - |
| CHEMBL1410134 | — | EC50 | > | 195000.0 | nM | - |
| CHEMBL1377188 | — | EC50 | > | 195000.0 | nM | - |
| CHEMBL1476311 | — | EC50 | > | 195000.0 | nM | - |
| CHEMBL1304057 | — | EC50 | > | 195000.0 | nM | - |