Assay Detail
Functional
CHEMBL1613892
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A screen for inhibitors of the PhoP region in Salmonella Typhi using a modified counterscreen. (Class of assay: confirmatory)
1028
Total Activities
1023
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1028 | 4.47 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1572266 | — | — | 1 | 6.46 |
| CHEMBL849 | TRICLOSAN | 4.0 | 1 | 6.43 |
| CHEMBL185 | FLUOROURACIL | 4.0 | 1 | 6.42 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | 4.0 | 1 | 6.42 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | -1.0 | 1 | 6.37 |
| CHEMBL1542959 | — | — | 1 | 6.36 |
| CHEMBL283849 | — | — | 1 | 6.35 |
| CHEMBL1587753 | — | — | 1 | 6.24 |
| CHEMBL22 | TRIMETHOPRIM | 4.0 | 1 | 6.17 |
| CHEMBL578512 | — | — | 1 | 6.13 |
| CHEMBL601757 | — | — | 1 | 6.11 |
| CHEMBL1594055 | — | — | 1 | 6.03 |
| CHEMBL1527664 | — | — | 1 | 5.96 |
| CHEMBL1326371 | — | — | 1 | 5.96 |
| CHEMBL1485275 | — | — | 1 | 5.93 |
| CHEMBL428064 | — | — | 1 | 5.93 |
| CHEMBL334707 | — | — | 1 | 5.84 |
| CHEMBL1593697 | — | — | 1 | 5.81 |
| CHEMBL1330220 | — | — | 1 | 5.76 |
| CHEMBL1513204 | — | — | 1 | 5.72 |
| CHEMBL1522007 | — | — | 1 | 5.71 |
| CHEMBL1200567 | — | — | 1 | 5.71 |
| CHEMBL1315061 | — | — | 1 | 5.68 |
| CHEMBL529 | AZITHROMYCIN | 4.0 | 1 | 5.63 |
| CHEMBL494760 | ORMETOPRIM | 2.0 | 1 | 5.62 |
| CHEMBL414400 | — | — | 1 | 5.59 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | — | 1 | 5.58 |
| CHEMBL130 | CHLORAMPHENICOL | 4.0 | 1 | 5.57 |
| CHEMBL1551640 | — | — | 1 | 5.53 |
| CHEMBL1329336 | — | — | 1 | 5.51 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1572266 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL849 | TRICLOSAN | IC50 | = | 369.0 | nM | 6.43 |
| CHEMBL185 | FLUOROURACIL | IC50 | = | 378.0 | nM | 6.42 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | IC50 | = | 376.0 | nM | 6.42 |
| CHEMBL1428564 | PEFLOXACIN MESYLATE | IC50 | = | 427.0 | nM | 6.37 |
| CHEMBL1542959 | — | IC50 | = | 441.0 | nM | 6.36 |
| CHEMBL283849 | — | IC50 | = | 444.0 | nM | 6.35 |
| CHEMBL1587753 | — | IC50 | = | 581.0 | nM | 6.24 |
| CHEMBL22 | TRIMETHOPRIM | IC50 | = | 675.0 | nM | 6.17 |
| CHEMBL578512 | — | IC50 | = | 741.0 | nM | 6.13 |
| CHEMBL601757 | — | IC50 | = | 781.0 | nM | 6.11 |
| CHEMBL1594055 | — | IC50 | = | 924.0 | nM | 6.03 |
| CHEMBL1326371 | — | IC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL1527664 | — | IC50 | = | 1096.0 | nM | 5.96 |
| CHEMBL428064 | — | IC50 | = | 1169.0 | nM | 5.93 |
| CHEMBL1485275 | — | IC50 | = | 1185.0 | nM | 5.93 |
| CHEMBL334707 | — | IC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL1593697 | — | IC50 | = | 1537.0 | nM | 5.81 |
| CHEMBL1330220 | — | IC50 | = | 1735.0 | nM | 5.76 |
| CHEMBL1513204 | — | IC50 | = | 1898.0 | nM | 5.72 |
| CHEMBL1200567 | — | IC50 | = | 1971.0 | nM | 5.71 |
| CHEMBL1522007 | — | IC50 | = | 1969.0 | nM | 5.71 |
| CHEMBL1315061 | — | IC50 | = | 2078.0 | nM | 5.68 |
| CHEMBL529 | AZITHROMYCIN | IC50 | = | 2334.0 | nM | 5.63 |
| CHEMBL494760 | ORMETOPRIM | IC50 | = | 2396.0 | nM | 5.62 |
| CHEMBL414400 | — | IC50 | = | 2553.0 | nM | 5.59 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | IC50 | = | 2609.0 | nM | 5.58 |
| CHEMBL130 | CHLORAMPHENICOL | IC50 | = | 2713.0 | nM | 5.57 |
| CHEMBL1551640 | — | IC50 | = | 2986.0 | nM | 5.53 |
| CHEMBL1329336 | — | IC50 | = | 3107.0 | nM | 5.51 |
| CHEMBL295619 | RUFLOXACIN | IC50 | = | 3158.0 | nM | 5.50 |
| CHEMBL1545940 | — | IC50 | = | 3206.0 | nM | 5.49 |
| CHEMBL1330113 | — | IC50 | = | 3245.0 | nM | 5.49 |
| CHEMBL1385206 | — | IC50 | = | 3492.0 | nM | 5.46 |
| CHEMBL1342852 | — | IC50 | = | 3547.0 | nM | 5.45 |
| CHEMBL1521960 | — | IC50 | = | 3618.0 | nM | 5.44 |
| CHEMBL290077 | — | IC50 | = | 3757.0 | nM | 5.42 |
| CHEMBL1330113 | — | IC50 | = | 3889.0 | nM | 5.41 |
| CHEMBL1456906 | — | IC50 | = | 4076.0 | nM | 5.39 |
| CHEMBL363449 | NADIFLOXACIN | IC50 | = | 4439.0 | nM | 5.35 |
| CHEMBL1327202 | — | IC50 | = | 4587.0 | nM | 5.34 |
| CHEMBL1241590 | FLORFENICOL | IC50 | = | 4739.0 | nM | 5.32 |
| CHEMBL139935 | — | IC50 | = | 4826.0 | nM | 5.32 |
| CHEMBL1385808 | — | IC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL1580272 | — | IC50 | = | 5092.0 | nM | 5.29 |
| CHEMBL790 | CHLORHEXIDINE | IC50 | = | 5354.0 | nM | 5.27 |
| CHEMBL1505275 | — | IC50 | = | 5643.0 | nM | 5.25 |
| CHEMBL727 | THIOGUANINE | IC50 | = | 6297.0 | nM | 5.20 |
| CHEMBL1378260 | — | IC50 | = | 6702.0 | nM | 5.17 |
| CHEMBL1441196 | — | IC50 | = | 7427.0 | nM | 5.13 |