Assay Detail
Functional
CHEMBL1613893
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: TR-FRET-based biochemical high throughput dose response assay for agonists of nuclear receptor subfamily 2, group E, member 3 (NR2E3). (Class of assay: confirmatory) [Related pubchem assays: 2379 (Screening (NR2E3 agonists, 3X)), 2325 (Summary), 2300 (Screening (NR2E3 agonists, 1X))]
125
Total Activities
125
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Photoreceptor-specific nuclear receptor (CHEMBL4374) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 125 | 5.83 | 6.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1391310 | — | — | 1 | 6.86 |
| CHEMBL1232381 | — | — | 1 | 6.83 |
| CHEMBL1575389 | — | — | 1 | 6.75 |
| CHEMBL1384281 | — | — | 1 | 6.75 |
| CHEMBL1326814 | — | — | 1 | 6.73 |
| CHEMBL1324779 | — | — | 1 | 6.66 |
| CHEMBL1544403 | — | — | 1 | 6.52 |
| CHEMBL1433074 | — | — | 1 | 6.48 |
| CHEMBL1454198 | — | — | 1 | 6.41 |
| CHEMBL1407788 | — | — | 1 | 6.00 |
| CHEMBL1391385 | — | — | 1 | 5.98 |
| CHEMBL1566010 | — | — | 1 | 5.96 |
| CHEMBL1499411 | — | — | 1 | 5.86 |
| CHEMBL1543331 | — | — | 1 | 5.85 |
| CHEMBL1536779 | — | — | 1 | 5.83 |
| CHEMBL1373811 | — | — | 1 | 5.79 |
| CHEMBL1580962 | — | — | 1 | 5.72 |
| CHEMBL1379684 | — | — | 1 | 5.69 |
| CHEMBL1336910 | — | — | 1 | 5.68 |
| CHEMBL1480178 | — | — | 1 | 5.63 |
| CHEMBL1549101 | — | — | 1 | 5.51 |
| CHEMBL1550435 | — | — | 1 | 5.42 |
| CHEMBL1369512 | — | — | 1 | 5.41 |
| CHEMBL1536665 | — | — | 1 | 5.39 |
| CHEMBL1501734 | — | — | 1 | 5.32 |
| CHEMBL1609827 | — | — | 1 | 5.29 |
| CHEMBL1592326 | — | — | 1 | 5.24 |
| CHEMBL1343308 | — | — | 1 | 5.24 |
| CHEMBL1462380 | — | — | 1 | 5.19 |
| CHEMBL1303255 | — | — | 1 | 5.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1391310 | — | IC50 | = | 139.1 | nM | 6.86 |
| CHEMBL1232381 | — | IC50 | = | 149.12 | nM | 6.83 |
| CHEMBL1384281 | — | IC50 | = | 177.87 | nM | 6.75 |
| CHEMBL1575389 | — | IC50 | = | 177.89 | nM | 6.75 |
| CHEMBL1326814 | — | IC50 | = | 185.5 | nM | 6.73 |
| CHEMBL1324779 | — | IC50 | = | 220.17 | nM | 6.66 |
| CHEMBL1544403 | — | IC50 | = | 303.35 | nM | 6.52 |
| CHEMBL1433074 | — | IC50 | = | 330.11 | nM | 6.48 |
| CHEMBL1454198 | — | IC50 | = | 389.38 | nM | 6.41 |
| CHEMBL1407788 | — | IC50 | = | 1001.0 | nM | 6.00 |
| CHEMBL1391385 | — | IC50 | = | 1056.0 | nM | 5.98 |
| CHEMBL1566010 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL1499411 | — | IC50 | = | 1378.0 | nM | 5.86 |
| CHEMBL1543331 | — | IC50 | = | 1421.0 | nM | 5.85 |
| CHEMBL1536779 | — | IC50 | = | 1492.0 | nM | 5.83 |
| CHEMBL1373811 | — | IC50 | = | 1636.0 | nM | 5.79 |
| CHEMBL1580962 | — | IC50 | = | 1903.0 | nM | 5.72 |
| CHEMBL1379684 | — | IC50 | = | 2039.0 | nM | 5.69 |
| CHEMBL1336910 | — | IC50 | = | 2092.0 | nM | 5.68 |
| CHEMBL1480178 | — | IC50 | = | 2320.0 | nM | 5.63 |
| CHEMBL1549101 | — | IC50 | = | 3055.0 | nM | 5.51 |
| CHEMBL1550435 | — | IC50 | = | 3837.0 | nM | 5.42 |
| CHEMBL1369512 | — | IC50 | = | 3852.0 | nM | 5.41 |
| CHEMBL1536665 | — | IC50 | = | 4111.0 | nM | 5.39 |
| CHEMBL1501734 | — | IC50 | = | 4746.0 | nM | 5.32 |
| CHEMBL1609827 | — | IC50 | = | 5106.0 | nM | 5.29 |
| CHEMBL1592326 | — | IC50 | = | 5733.0 | nM | 5.24 |
| CHEMBL1343308 | — | IC50 | = | 5775.0 | nM | 5.24 |
| CHEMBL1462380 | — | IC50 | = | 6407.0 | nM | 5.19 |
| CHEMBL1303255 | — | IC50 | = | 8407.0 | nM | 5.08 |
| CHEMBL1455509 | — | IC50 | = | 12372.0 | nM | 4.91 |
| CHEMBL1386595 | — | IC50 | = | 32959.0 | nM | 4.48 |
| CHEMBL1511291 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1427088 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1347701 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1432707 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1505221 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1353643 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1565261 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1307313 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1307433 | — | IC50 | > | 1476.0 | nM | - |
| CHEMBL1388002 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1600749 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1573867 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1601179 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL578512 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL388590 | BENZBROMARONE | IC50 | > | 39841.0 | nM | - |
| CHEMBL1535636 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1601448 | — | IC50 | > | 39841.0 | nM | - |
| CHEMBL1569119 | — | IC50 | > | 39841.0 | nM | - |