Assay Detail
Functional
CHEMBL1613956
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response counterscreen for neuropeptide Y receptor Y2 (NPY-Y2): Cell-based high throughput assay to measure NPY-Y1 antagonism. (Class of assay: confirmatory) [Related pubchem assays: 1256, 793, 1257 ]
119
Total Activities
119
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 119 | 5.12 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1345334 | — | — | 1 | 5.40 |
| CHEMBL1428935 | — | — | 1 | 5.39 |
| CHEMBL1353428 | — | — | 1 | 5.39 |
| CHEMBL1402158 | — | — | 1 | 5.37 |
| CHEMBL1502859 | — | — | 1 | 5.36 |
| CHEMBL1312713 | — | — | 1 | 5.36 |
| CHEMBL1580409 | — | — | 1 | 5.35 |
| CHEMBL417727 | — | — | 1 | 5.34 |
| CHEMBL1531745 | — | — | 1 | 5.34 |
| CHEMBL1419096 | — | — | 1 | 5.32 |
| CHEMBL1471779 | — | — | 1 | 5.32 |
| CHEMBL1499276 | — | — | 1 | 5.30 |
| CHEMBL3211272 | — | — | 1 | 5.30 |
| CHEMBL1468302 | — | — | 1 | 5.29 |
| CHEMBL1585445 | — | — | 1 | 5.29 |
| CHEMBL1457093 | — | — | 1 | 5.29 |
| CHEMBL1201049 | ECONAZOLE NITRATE | 4.0 | 1 | 5.29 |
| CHEMBL1559259 | — | — | 1 | 5.28 |
| CHEMBL1522356 | — | — | 1 | 5.28 |
| CHEMBL1427745 | — | — | 1 | 5.28 |
| CHEMBL1312703 | — | — | 1 | 5.28 |
| CHEMBL1537995 | — | — | 1 | 5.27 |
| CHEMBL3195229 | — | — | 1 | 5.27 |
| CHEMBL1308845 | — | — | 1 | 5.27 |
| CHEMBL1568243 | — | — | 1 | 5.26 |
| CHEMBL1348426 | — | — | 1 | 5.26 |
| CHEMBL1431004 | — | — | 1 | 5.26 |
| CHEMBL1423799 | — | — | 1 | 5.25 |
| CHEMBL1427504 | — | — | 1 | 5.25 |
| CHEMBL1487131 | — | — | 1 | 5.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1345334 | — | IC50 | = | 4021.0 | nM | 5.40 |
| CHEMBL1353428 | — | IC50 | = | 4084.0 | nM | 5.39 |
| CHEMBL1428935 | — | IC50 | = | 4079.0 | nM | 5.39 |
| CHEMBL1402158 | — | IC50 | = | 4261.0 | nM | 5.37 |
| CHEMBL1312713 | — | IC50 | = | 4368.0 | nM | 5.36 |
| CHEMBL1502859 | — | IC50 | = | 4380.0 | nM | 5.36 |
| CHEMBL1580409 | — | IC50 | = | 4465.0 | nM | 5.35 |
| CHEMBL417727 | — | IC50 | = | 4542.0 | nM | 5.34 |
| CHEMBL1531745 | — | IC50 | = | 4576.0 | nM | 5.34 |
| CHEMBL1471779 | — | IC50 | = | 4838.0 | nM | 5.32 |
| CHEMBL1419096 | — | IC50 | = | 4826.0 | nM | 5.32 |
| CHEMBL1499276 | — | IC50 | = | 5010.0 | nM | 5.30 |
| CHEMBL3211272 | — | IC50 | = | 5022.0 | nM | 5.30 |
| CHEMBL1468302 | — | IC50 | = | 5100.0 | nM | 5.29 |
| CHEMBL1201049 | ECONAZOLE NITRATE | IC50 | = | 5146.0 | nM | 5.29 |
| CHEMBL1457093 | — | IC50 | = | 5161.0 | nM | 5.29 |
| CHEMBL1585445 | — | IC50 | = | 5137.0 | nM | 5.29 |
| CHEMBL1312703 | — | IC50 | = | 5306.0 | nM | 5.28 |
| CHEMBL1427745 | — | IC50 | = | 5265.0 | nM | 5.28 |
| CHEMBL1522356 | — | IC50 | = | 5266.0 | nM | 5.28 |
| CHEMBL1559259 | — | IC50 | = | 5210.0 | nM | 5.28 |
| CHEMBL1537995 | — | IC50 | = | 5404.0 | nM | 5.27 |
| CHEMBL1308845 | — | IC50 | = | 5388.0 | nM | 5.27 |
| CHEMBL3195229 | — | IC50 | = | 5335.0 | nM | 5.27 |
| CHEMBL1568243 | — | IC50 | = | 5470.0 | nM | 5.26 |
| CHEMBL1348426 | — | IC50 | = | 5546.0 | nM | 5.26 |
| CHEMBL1431004 | — | IC50 | = | 5537.0 | nM | 5.26 |
| CHEMBL1487131 | — | IC50 | = | 5680.0 | nM | 5.25 |
| CHEMBL1427504 | — | IC50 | = | 5687.0 | nM | 5.25 |
| CHEMBL1423799 | — | IC50 | = | 5687.0 | nM | 5.25 |
| CHEMBL1453672 | — | IC50 | = | 5724.0 | nM | 5.24 |
| CHEMBL1493500 | — | IC50 | = | 5769.0 | nM | 5.24 |
| CHEMBL1426896 | — | IC50 | = | 5853.0 | nM | 5.23 |
| CHEMBL1310577 | — | IC50 | = | 6031.0 | nM | 5.22 |
| CHEMBL1335124 | — | IC50 | = | 6127.0 | nM | 5.21 |
| CHEMBL1379143 | — | IC50 | = | 6324.0 | nM | 5.20 |
| CHEMBL3190644 | — | IC50 | = | 6459.0 | nM | 5.19 |
| CHEMBL1393538 | — | IC50 | = | 6433.0 | nM | 5.19 |
| CHEMBL1327690 | — | IC50 | = | 6664.0 | nM | 5.18 |
| CHEMBL1574689 | — | IC50 | = | 6952.0 | nM | 5.16 |
| CHEMBL1610409 | — | IC50 | = | 6959.0 | nM | 5.16 |
| CHEMBL1446166 | — | IC50 | = | 6943.0 | nM | 5.16 |
| CHEMBL1545971 | — | IC50 | = | 7125.0 | nM | 5.15 |
| CHEMBL1990096 | — | IC50 | = | 7084.0 | nM | 5.15 |
| CHEMBL3208997 | — | IC50 | = | 7083.0 | nM | 5.15 |
| CHEMBL1308461 | — | IC50 | = | 7229.0 | nM | 5.14 |
| CHEMBL564979 | — | IC50 | = | 7273.0 | nM | 5.14 |
| CHEMBL1480648 | — | IC50 | = | 7156.0 | nM | 5.14 |
| CHEMBL1311570 | — | IC50 | = | 7444.0 | nM | 5.13 |
| CHEMBL1383592 | — | IC50 | = | 7387.0 | nM | 5.13 |