Assay Detail
Functional
CHEMBL1614047
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: PMA/Ionomycin induced NF-kB luciferase assay in 293- NF-kB-Luc stable cells. (Class of assay: confirmatory) [Related pubchem assays: 1299, 1270, 1295, 1375, 1287, 1281, 1293, 1291, 1289, 1280, 465, 1364, 1282, 1372, 1365, 1370, 1367, 1366, 1269, 1373, 1292, 1290, 1302, 1371, 1283, 1271, 1294, 1374, 1368, 1369 ]
28
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 28 | 5.74 | 7.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1579491 | — | — | 1 | 7.26 |
| CHEMBL1427791 | — | — | 1 | 6.89 |
| CHEMBL1576870 | — | — | 1 | 6.35 |
| CHEMBL1370087 | — | — | 1 | 6.34 |
| CHEMBL1403324 | — | — | 1 | 6.28 |
| CHEMBL1170624 | — | — | 1 | 6.19 |
| CHEMBL1579418 | — | — | 1 | 6.13 |
| CHEMBL1372889 | — | — | 1 | 6.11 |
| CHEMBL1566033 | — | — | 1 | 6.11 |
| CHEMBL1589625 | — | — | 1 | 6.00 |
| CHEMBL1401969 | — | — | 1 | 5.93 |
| CHEMBL42529 | — | — | 2 | 5.73 |
| CHEMBL373137 | — | — | 1 | 5.66 |
| CHEMBL1172202 | — | — | 1 | 5.56 |
| CHEMBL1491842 | — | — | 1 | 5.56 |
| CHEMBL1611128 | — | — | 1 | 5.56 |
| CHEMBL1557774 | — | — | 1 | 5.48 |
| CHEMBL1410813 | — | — | 1 | 5.38 |
| CHEMBL1410454 | — | — | 1 | 5.38 |
| CHEMBL1482541 | — | — | 1 | 5.37 |
| CHEMBL363657 | — | — | 1 | 5.37 |
| CHEMBL1504484 | — | — | 1 | 5.21 |
| CHEMBL1600399 | — | — | 1 | 5.01 |
| CHEMBL1518672 | — | — | 1 | 4.90 |
| CHEMBL1578584 | — | — | 1 | 4.81 |
| CHEMBL1309478 | — | — | 1 | 4.80 |
| CHEMBL1407693 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1579491 | — | EC50 | = | 55.18 | nM | 7.26 |
| CHEMBL1427791 | — | EC50 | = | 128.6 | nM | 6.89 |
| CHEMBL1576870 | — | EC50 | = | 443.4 | nM | 6.35 |
| CHEMBL1370087 | — | EC50 | = | 456.1 | nM | 6.34 |
| CHEMBL1403324 | — | EC50 | = | 529.5 | nM | 6.28 |
| CHEMBL1170624 | — | EC50 | = | 643.9 | nM | 6.19 |
| CHEMBL1579418 | — | EC50 | = | 743.8 | nM | 6.13 |
| CHEMBL1566033 | — | EC50 | = | 781.4 | nM | 6.11 |
| CHEMBL1372889 | — | EC50 | = | 773.5 | nM | 6.11 |
| CHEMBL1589625 | — | EC50 | = | 1003.0 | nM | 6.00 |
| CHEMBL1401969 | — | EC50 | = | 1168.0 | nM | 5.93 |
| CHEMBL42529 | — | EC50 | = | 1846.0 | nM | 5.73 |
| CHEMBL42529 | — | EC50 | = | 1846.0 | nM | 5.73 |
| CHEMBL373137 | — | EC50 | = | 2177.0 | nM | 5.66 |
| CHEMBL1172202 | — | EC50 | = | 2776.0 | nM | 5.56 |
| CHEMBL1491842 | — | EC50 | = | 2767.0 | nM | 5.56 |
| CHEMBL1611128 | — | EC50 | = | 2770.0 | nM | 5.56 |
| CHEMBL1557774 | — | EC50 | = | 3290.0 | nM | 5.48 |
| CHEMBL1410813 | — | EC50 | = | 4206.0 | nM | 5.38 |
| CHEMBL1410454 | — | EC50 | = | 4194.0 | nM | 5.38 |
| CHEMBL1482541 | — | EC50 | = | 4251.0 | nM | 5.37 |
| CHEMBL363657 | — | EC50 | = | 4243.0 | nM | 5.37 |
| CHEMBL1504484 | — | EC50 | = | 6118.0 | nM | 5.21 |
| CHEMBL1600399 | — | EC50 | = | 9821.0 | nM | 5.01 |
| CHEMBL1518672 | — | EC50 | = | 12520.0 | nM | 4.90 |
| CHEMBL1578584 | — | EC50 | = | 15430.0 | nM | 4.81 |
| CHEMBL1309478 | — | EC50 | = | 15750.0 | nM | 4.80 |
| CHEMBL1407693 | — | EC50 | < | 4000.0 | nM | - |