Assay Detail
Binding
CHEMBL1614063
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PUBCHEM_BIOASSAY: GAPDH Dose Response Colorimetric Assay. (Class of assay: confirmatory)
744
Total Activities
744
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Glyceraldehyde-3-phosphate dehydrogenase (CHEMBL2284) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 744 | 4.29 | 5.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1371869 | — | — | 1 | 5.64 |
| CHEMBL1452781 | — | — | 1 | 5.28 |
| CHEMBL502775 | — | — | 1 | 4.80 |
| CHEMBL1603381 | — | — | 1 | 4.56 |
| CHEMBL1526610 | — | — | 1 | 4.56 |
| CHEMBL1427609 | — | — | 1 | 4.56 |
| CHEMBL201289 | — | — | 1 | 4.54 |
| CHEMBL1319947 | — | — | 1 | 4.44 |
| CHEMBL1430473 | — | — | 1 | 4.42 |
| CHEMBL1527520 | — | — | 1 | 4.32 |
| CHEMBL1363132 | — | — | 1 | 4.32 |
| CHEMBL1403754 | — | — | 1 | 4.30 |
| CHEMBL1452440 | — | — | 1 | 4.25 |
| CHEMBL1409373 | — | — | 1 | 4.21 |
| CHEMBL1328398 | — | — | 1 | 4.20 |
| CHEMBL1608225 | — | — | 1 | 4.20 |
| CHEMBL1376870 | — | — | 1 | 4.15 |
| CHEMBL1608153 | — | — | 1 | 4.12 |
| CHEMBL1570803 | — | — | 1 | 4.12 |
| CHEMBL1447034 | — | — | 1 | 4.09 |
| CHEMBL1374971 | — | — | 1 | 4.09 |
| CHEMBL1373046 | — | — | 1 | 4.06 |
| CHEMBL1608654 | — | — | 1 | 4.06 |
| CHEMBL1528814 | — | — | 1 | 4.05 |
| CHEMBL578585 | — | — | 1 | 4.04 |
| CHEMBL1334412 | — | — | 1 | 4.04 |
| CHEMBL1386069 | — | — | 1 | 4.03 |
| CHEMBL1606543 | — | — | 1 | 4.03 |
| CHEMBL1334633 | — | — | 1 | 4.02 |
| CHEMBL1353227 | — | — | 1 | 4.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1371869 | — | IC50 | = | 2310.0 | nM | 5.64 |
| CHEMBL1452781 | — | IC50 | = | 5300.0 | nM | 5.28 |
| CHEMBL502775 | — | IC50 | = | 15800.0 | nM | 4.80 |
| CHEMBL1526610 | — | IC50 | = | 27400.0 | nM | 4.56 |
| CHEMBL1427609 | — | IC50 | = | 27400.0 | nM | 4.56 |
| CHEMBL1603381 | — | IC50 | = | 27800.0 | nM | 4.56 |
| CHEMBL201289 | — | IC50 | = | 28700.0 | nM | 4.54 |
| CHEMBL1319947 | — | IC50 | = | 36300.0 | nM | 4.44 |
| CHEMBL1430473 | — | IC50 | = | 37800.0 | nM | 4.42 |
| CHEMBL1363132 | — | IC50 | = | 47800.0 | nM | 4.32 |
| CHEMBL1527520 | — | IC50 | = | 47700.0 | nM | 4.32 |
| CHEMBL1403754 | — | IC50 | = | 50100.0 | nM | 4.30 |
| CHEMBL1452440 | — | IC50 | = | 56400.0 | nM | 4.25 |
| CHEMBL1409373 | — | IC50 | = | 62200.0 | nM | 4.21 |
| CHEMBL1608225 | — | IC50 | = | 62700.0 | nM | 4.20 |
| CHEMBL1328398 | — | IC50 | = | 62600.0 | nM | 4.20 |
| CHEMBL1376870 | — | IC50 | = | 70700.0 | nM | 4.15 |
| CHEMBL1608153 | — | IC50 | = | 76800.0 | nM | 4.12 |
| CHEMBL1570803 | — | IC50 | = | 76600.0 | nM | 4.12 |
| CHEMBL1447034 | — | IC50 | = | 80800.0 | nM | 4.09 |
| CHEMBL1374971 | — | IC50 | = | 81200.0 | nM | 4.09 |
| CHEMBL1373046 | — | IC50 | = | 87300.0 | nM | 4.06 |
| CHEMBL1608654 | — | IC50 | = | 87100.0 | nM | 4.06 |
| CHEMBL1528814 | — | IC50 | = | 88900.0 | nM | 4.05 |
| CHEMBL1334412 | — | IC50 | = | 91400.0 | nM | 4.04 |
| CHEMBL578585 | — | IC50 | = | 92200.0 | nM | 4.04 |
| CHEMBL1606543 | — | IC50 | = | 93600.0 | nM | 4.03 |
| CHEMBL1386069 | — | IC50 | = | 93800.0 | nM | 4.03 |
| CHEMBL1334633 | — | IC50 | = | 95400.0 | nM | 4.02 |
| CHEMBL1353227 | — | IC50 | = | 98600.0 | nM | 4.01 |
| CHEMBL1570401 | — | IC50 | = | 97400.0 | nM | 4.01 |
| CHEMBL1449334 | — | IC50 | = | 99100.0 | nM | 4.00 |
| CHEMBL1492839 | — | IC50 | = | 99700.0 | nM | 4.00 |
| CHEMBL1372161 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL466809 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL178453 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1450886 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1535015 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1326265 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL442458 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1490393 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1495968 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1405375 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1490321 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1411988 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1412561 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1412060 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL315708 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1412224 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1523213 | — | IC50 | > | 100000.0 | nM | - |