Assay Detail
Functional
CHEMBL1614065
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response to Identify Inhibitors of 5'UTR Stem-Loop Driven Prion Protein mRNA Translation in H4-C Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1827 (Project Summary), 1813 (Primary HTS)]
183
Total Activities
183
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 183 | 6.35 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1462938 | — | — | 1 | 7.92 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 7.85 |
| CHEMBL1555935 | — | — | 1 | 7.80 |
| CHEMBL1562575 | — | — | 1 | 7.68 |
| CHEMBL3192138 | — | — | 1 | 7.58 |
| CHEMBL1536981 | — | — | 1 | 7.57 |
| CHEMBL3195389 | — | — | 1 | 7.44 |
| CHEMBL1751 | DIGOXIN | 4.0 | 1 | 7.40 |
| CHEMBL1342336 | — | — | 1 | 7.34 |
| CHEMBL1368103 | — | — | 1 | 7.22 |
| CHEMBL501867 | VINCRISTINE SULFATE | 4.0 | 1 | 7.20 |
| CHEMBL300389 | — | — | 1 | 7.12 |
| CHEMBL3185655 | — | — | 1 | 7.12 |
| CHEMBL1884996 | — | — | 1 | 7.12 |
| CHEMBL1376974 | — | — | 1 | 7.11 |
| CHEMBL1987060 | — | — | 1 | 7.11 |
| CHEMBL222863 | OUABAIN | -1.0 | 1 | 7.10 |
| CHEMBL1355541 | — | — | 1 | 7.10 |
| CHEMBL312862 | DEMECOLCINE | 2.0 | 1 | 7.10 |
| CHEMBL1312738 | — | — | 1 | 7.08 |
| CHEMBL290077 | — | — | 1 | 7.08 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.07 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | -1.0 | 1 | 7.00 |
| CHEMBL513000 | — | — | 1 | 7.00 |
| CHEMBL1602385 | — | — | 1 | 7.00 |
| CHEMBL1587117 | — | — | 1 | 7.00 |
| CHEMBL1595169 | — | — | 1 | 6.98 |
| CHEMBL460601 | — | — | 1 | 6.95 |
| CHEMBL373137 | — | — | 1 | 6.94 |
| CHEMBL1347346 | — | — | 1 | 6.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1462938 | — | EC50 | = | 12.0 | nM | 7.92 |
| CHEMBL61 | PODOFILOX | EC50 | = | 14.0 | nM | 7.85 |
| CHEMBL1555935 | — | EC50 | = | 16.0 | nM | 7.80 |
| CHEMBL1562575 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL3192138 | — | EC50 | = | 26.0 | nM | 7.58 |
| CHEMBL1536981 | — | EC50 | = | 27.0 | nM | 7.57 |
| CHEMBL3195389 | — | EC50 | = | 36.0 | nM | 7.44 |
| CHEMBL1751 | DIGOXIN | EC50 | = | 40.0 | nM | 7.40 |
| CHEMBL1342336 | — | EC50 | = | 46.0 | nM | 7.34 |
| CHEMBL1368103 | — | EC50 | = | 60.0 | nM | 7.22 |
| CHEMBL501867 | VINCRISTINE SULFATE | EC50 | = | 63.0 | nM | 7.20 |
| CHEMBL3185655 | — | EC50 | = | 75.0 | nM | 7.12 |
| CHEMBL1884996 | — | EC50 | = | 76.0 | nM | 7.12 |
| CHEMBL300389 | — | EC50 | = | 76.0 | nM | 7.12 |
| CHEMBL1987060 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1376974 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1355541 | — | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL222863 | OUABAIN | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL312862 | DEMECOLCINE | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL290077 | — | EC50 | = | 84.0 | nM | 7.08 |
| CHEMBL1312738 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL428647 | PACLITAXEL | EC50 | = | 86.0 | nM | 7.07 |
| CHEMBL1602385 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1587117 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL513000 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1595169 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL460601 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL373137 | — | EC50 | = | 116.0 | nM | 6.94 |
| CHEMBL1347346 | — | EC50 | = | 114.0 | nM | 6.94 |
| CHEMBL423192 | ANISOMYCIN | EC50 | = | 121.0 | nM | 6.92 |
| CHEMBL1453996 | — | EC50 | = | 123.0 | nM | 6.91 |
| CHEMBL1372889 | — | EC50 | = | 135.0 | nM | 6.87 |
| CHEMBL1392142 | — | EC50 | = | 146.0 | nM | 6.84 |
| CHEMBL1323774 | — | EC50 | = | 163.0 | nM | 6.79 |
| CHEMBL1307091 | — | EC50 | = | 178.0 | nM | 6.75 |
| CHEMBL1540099 | — | EC50 | = | 179.0 | nM | 6.75 |
| CHEMBL1473676 | — | EC50 | = | 190.0 | nM | 6.72 |
| CHEMBL1495092 | — | EC50 | = | 194.0 | nM | 6.71 |
| CHEMBL9514 | NOCODAZOLE | EC50 | = | 203.0 | nM | 6.69 |
| CHEMBL1528660 | — | EC50 | = | 215.0 | nM | 6.67 |
| CHEMBL267099 | TUBERCIDIN | EC50 | = | 223.0 | nM | 6.65 |
| CHEMBL304291 | — | EC50 | = | 222.0 | nM | 6.65 |
| CHEMBL1405749 | — | EC50 | = | 229.0 | nM | 6.64 |
| CHEMBL1537509 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1316831 | — | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL222409 | — | EC50 | = | 233.0 | nM | 6.63 |
| CHEMBL579318 | — | EC50 | = | 232.0 | nM | 6.63 |
| CHEMBL1479301 | — | EC50 | = | 253.0 | nM | 6.60 |
| CHEMBL1432507 | — | EC50 | = | 255.0 | nM | 6.59 |