Assay Detail
Functional
CHEMBL1614105
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: AlphaScreen confirmatory assay for validation of inhibitors of SUMOylation. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2006, AID2011, AID2069, AID2614, AID2658]
327
Total Activities
327
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 327 | 5.10 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3190558 | — | — | 1 | 6.46 |
| CHEMBL1598762 | — | — | 1 | 6.38 |
| CHEMBL1401747 | — | — | 1 | 6.28 |
| CHEMBL1518098 | — | — | 1 | 6.27 |
| CHEMBL33864 | LIPOIC ACID, ALPHA | 3.0 | 1 | 6.21 |
| CHEMBL1405964 | — | — | 1 | 6.17 |
| CHEMBL3196108 | — | — | 1 | 6.17 |
| CHEMBL1997990 | — | — | 1 | 6.16 |
| CHEMBL1985987 | — | — | 1 | 6.13 |
| CHEMBL1530147 | — | — | 1 | 6.07 |
| CHEMBL1426692 | — | — | 1 | 6.07 |
| CHEMBL1612112 | — | — | 1 | 6.06 |
| CHEMBL1376540 | — | — | 1 | 6.06 |
| CHEMBL1575869 | — | — | 1 | 6.05 |
| CHEMBL1529471 | — | — | 1 | 6.01 |
| CHEMBL3189845 | — | — | 1 | 6.00 |
| CHEMBL1582771 | — | — | 1 | 6.00 |
| CHEMBL3195531 | — | — | 1 | 6.00 |
| CHEMBL1427775 | — | — | 1 | 5.96 |
| CHEMBL1522941 | — | — | 1 | 5.95 |
| CHEMBL1508847 | — | — | 1 | 5.95 |
| CHEMBL1091723 | — | — | 1 | 5.94 |
| CHEMBL1307317 | — | — | 1 | 5.93 |
| CHEMBL1418005 | — | — | 1 | 5.92 |
| CHEMBL3214310 | — | — | 1 | 5.92 |
| CHEMBL1488474 | — | — | 1 | 5.90 |
| CHEMBL1996724 | — | — | 1 | 5.87 |
| CHEMBL2000877 | — | — | 1 | 5.86 |
| CHEMBL1340834 | — | — | 1 | 5.86 |
| CHEMBL1874620 | — | — | 1 | 5.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3190558 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL1598762 | — | IC50 | = | 420.0 | nM | 6.38 |
| CHEMBL1401747 | — | IC50 | = | 530.0 | nM | 6.28 |
| CHEMBL1518098 | — | IC50 | = | 540.0 | nM | 6.27 |
| CHEMBL33864 | LIPOIC ACID, ALPHA | IC50 | = | 620.0 | nM | 6.21 |
| CHEMBL1405964 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL3196108 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1997990 | — | IC50 | = | 690.0 | nM | 6.16 |
| CHEMBL1985987 | — | IC50 | = | 740.0 | nM | 6.13 |
| CHEMBL1530147 | — | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL1426692 | — | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL1612112 | — | IC50 | = | 880.0 | nM | 6.06 |
| CHEMBL1376540 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL1575869 | — | IC50 | = | 890.0 | nM | 6.05 |
| CHEMBL1529471 | — | IC50 | = | 980.0 | nM | 6.01 |
| CHEMBL3195531 | — | IC50 | = | 990.0 | nM | 6.00 |
| CHEMBL1582771 | — | IC50 | = | 990.0 | nM | 6.00 |
| CHEMBL3189845 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1427775 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL1522941 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1508847 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1091723 | — | IC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL1307317 | — | IC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL1418005 | — | IC50 | = | 1210.0 | nM | 5.92 |
| CHEMBL3214310 | — | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL1488474 | — | IC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1996724 | — | IC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL1340834 | — | IC50 | = | 1390.0 | nM | 5.86 |
| CHEMBL2000877 | — | IC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL1874620 | — | IC50 | = | 1410.0 | nM | 5.85 |
| CHEMBL1561488 | — | IC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL299853 | — | IC50 | = | 1470.0 | nM | 5.83 |
| CHEMBL1966168 | — | IC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1446626 | — | IC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1888528 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL1461225 | — | IC50 | = | 1580.0 | nM | 5.80 |
| CHEMBL3212364 | — | IC50 | = | 1640.0 | nM | 5.79 |
| CHEMBL1481301 | — | IC50 | = | 1620.0 | nM | 5.79 |
| CHEMBL1520133 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL1255778 | BENSERAZIDE HYDROCHLORIDE | IC50 | = | 1660.0 | nM | 5.78 |
| CHEMBL1993780 | — | IC50 | = | 1710.0 | nM | 5.77 |
| CHEMBL1522351 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL1379448 | — | IC50 | = | 1820.0 | nM | 5.74 |
| CHEMBL1516834 | — | IC50 | = | 1840.0 | nM | 5.74 |
| CHEMBL1503523 | — | IC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL2005973 | — | IC50 | = | 1860.0 | nM | 5.73 |
| CHEMBL3194086 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1495592 | — | IC50 | = | 2060.0 | nM | 5.69 |
| CHEMBL175434 | — | IC50 | = | 2110.0 | nM | 5.68 |
| CHEMBL1312212 | — | IC50 | = | 2150.0 | nM | 5.67 |