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Assay Detail

CHEMBL1614151

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: A Cell Based HTS Approach for the Discovery of New Inhibitors of Respiratory syncytial virus (RSV). (Class of assay: confirmatory)
409
Total Activities
409
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 409 4.82 6.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1433302 1 6.28
CHEMBL1378226 1 6.24
CHEMBL1382599 1 6.00
CHEMBL1588704 1 5.96
CHEMBL3209968 1 5.94
CHEMBL3213457 1 5.94
CHEMBL1548010 1 5.91
CHEMBL1520067 1 5.90
CHEMBL1542320 1 5.84
CHEMBL1579405 1 5.83
CHEMBL1528707 1 5.82
CHEMBL3209011 1 5.75
CHEMBL1495736 1 5.73
CHEMBL1464327 1 5.72
CHEMBL3194919 1 5.72
CHEMBL1483754 1 5.70
CHEMBL564201 6-AZAURIDINE 1 5.64
CHEMBL1574420 1 5.62
CHEMBL1459342 1 5.61
CHEMBL3211659 1 5.59
CHEMBL1502132 1 5.59
CHEMBL3213449 1 5.58
CHEMBL1467286 1 5.55
CHEMBL1580974 1 5.54
CHEMBL1526941 1 5.53
CHEMBL1359367 1 5.51
CHEMBL1353865 1 5.51
CHEMBL1446667 1 5.50
CHEMBL1330929 1 5.48
CHEMBL1426851 1 5.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1433302 IC50 = 530.0 nM 6.28
CHEMBL1378226 IC50 = 580.0 nM 6.24
CHEMBL1382599 IC50 = 1010.0 nM 6.00
CHEMBL1588704 IC50 = 1100.0 nM 5.96
CHEMBL3209968 IC50 = 1140.0 nM 5.94
CHEMBL3213457 IC50 = 1140.0 nM 5.94
CHEMBL1548010 IC50 = 1220.0 nM 5.91
CHEMBL1520067 IC50 = 1260.0 nM 5.90
CHEMBL1542320 IC50 = 1430.0 nM 5.84
CHEMBL1579405 IC50 = 1470.0 nM 5.83
CHEMBL1528707 IC50 = 1530.0 nM 5.82
CHEMBL3209011 IC50 = 1770.0 nM 5.75
CHEMBL1495736 IC50 = 1860.0 nM 5.73
CHEMBL1464327 IC50 = 1910.0 nM 5.72
CHEMBL3194919 IC50 = 1910.0 nM 5.72
CHEMBL1483754 IC50 = 2020.0 nM 5.70
CHEMBL564201 6-AZAURIDINE IC50 = 2280.0 nM 5.64
CHEMBL1574420 IC50 = 2400.0 nM 5.62
CHEMBL1459342 IC50 = 2480.0 nM 5.61
CHEMBL1502132 IC50 = 2540.0 nM 5.59
CHEMBL3211659 IC50 = 2580.0 nM 5.59
CHEMBL3213449 IC50 = 2620.0 nM 5.58
CHEMBL1467286 IC50 = 2830.0 nM 5.55
CHEMBL1580974 IC50 = 2910.0 nM 5.54
CHEMBL1526941 IC50 = 2980.0 nM 5.53
CHEMBL1359367 IC50 = 3120.0 nM 5.51
CHEMBL1353865 IC50 = 3070.0 nM 5.51
CHEMBL1446667 IC50 = 3140.0 nM 5.50
CHEMBL1330929 IC50 = 3310.0 nM 5.48
CHEMBL1426851 IC50 = 3340.0 nM 5.48
CHEMBL1452228 IC50 = 3400.0 nM 5.47
CHEMBL1374924 IC50 = 3550.0 nM 5.45
CHEMBL1550640 IC50 = 3580.0 nM 5.45
CHEMBL1538446 IC50 = 3600.0 nM 5.44
CHEMBL1526395 IC50 = 3620.0 nM 5.44
CHEMBL1546303 IC50 = 3750.0 nM 5.43
CHEMBL1599784 IC50 = 3980.0 nM 5.40
CHEMBL1474104 IC50 = 4070.0 nM 5.39
CHEMBL1528529 IC50 = 4080.0 nM 5.39
CHEMBL1402135 IC50 = 4180.0 nM 5.38
CHEMBL1474991 IC50 = 4370.0 nM 5.36
CHEMBL1392893 IC50 = 4490.0 nM 5.35
CHEMBL1408835 IC50 = 4430.0 nM 5.35
CHEMBL1378307 IC50 = 4510.0 nM 5.35
CHEMBL1412578 IC50 = 4570.0 nM 5.34
CHEMBL1359923 IC50 = 4690.0 nM 5.33
CHEMBL1311916 IC50 = 4720.0 nM 5.33
CHEMBL1310551 IC50 = 4820.0 nM 5.32
CHEMBL1497106 IC50 = 4750.0 nM 5.32
CHEMBL1594943 IC50 = 4770.0 nM 5.32