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Compound Detail

CHEMBL1495736

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Cc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2cccc3cccnc23)c(C)c1

Basic Information

ChEMBL ID CHEMBL1495736
Phase Preclinical
Structure Type MOL
InChI Key DWDDBDJWOXJEMQ-UHFFFAOYSA-N
2
Targets
2
Activities
2
Assay Types
0
PK Parameters
3
Publications
0
Known Names

Molecular Properties

409.5
MW (Da)
3.64
ALogP
4
HBA
1
HBD
79.4
PSA (Ų)
0.71
QED
0
Ro5 Violations
4
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C22H23N3O3S
MW 409.51
Aromatic Rings 3
Heavy Atoms 29
NP-Likeness -2.09

Activity Summary

EC50 1 meas. best 5.3
IC50 1 meas. best 5.73

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.73 5.73 1860.0 1
Respiratory syncytial virus
CHEMBL612679
EC50 5.3 5.3 5000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
23043370 10.1021/jm300612z Respiratory syncytial virus 2
23043370 10.1021/jm300612z Unchecked 1
23043370 10.1021/jm300612z HEp-2 1

Data from ChEMBL 36 via Core Engine