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Compound Detail

CHEMBL1520067

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Cc1cccc(-n2c(SCC(=O)Nc3ncc(Cl)cc3Cl)nc3ccccc32)c1

Basic Information

ChEMBL ID CHEMBL1520067
Phase Preclinical
Structure Type MOL
InChI Key MMKPVKCGCNPSQC-UHFFFAOYSA-N
3
Targets
5
Activities
2
Assay Types
0
PK Parameters
1
Publications
0
Known Names

Molecular Properties

443.4
MW (Da)
5.77
ALogP
5
HBA
1
HBD
59.8
PSA (Ų)
0.40
QED
1
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C21H16Cl2N4OS
MW 443.36
Aromatic Rings 4
Heavy Atoms 29
NP-Likeness -2.62

Activity Summary

EC50 4 meas. best 5.68
IC50 1 meas. best 5.9

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 5.9 5.9 1260.0 1
Measles morbillivirus
CHEMBL613738
EC50 5.68 5.68 2100.0 1
BJ
CHEMBL614358
EC50 4.47 4.385 33690.0 2
Unchecked
CHEMBL612545
EC50 4.03 4.03 94193.0 1

Activity Data Samples

Top measurements by pChEMBL value

Literature References

PubMed DOI Target Context # Activities
22328961 10.1021/ml200125r Measles morbillivirus 1

Data from ChEMBL 36 via Core Engine