Assay Detail
Functional
CHEMBL1614155
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Confirmation HTS to Identify Compounds Cytotoxic to BJeLR RAS-Dependent Fibroblast. (Class of assay: confirmatory) [Related pubchem assays: 1674 (Project Summary), 1554 (Primary HTS)]
1153
Total Activities
1153
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | BJ |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1153 | 5.10 | 6.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL323668 | — | — | 1 | 6.90 |
| CHEMBL225071 | RALTITREXED | 4.0 | 1 | 6.72 |
| CHEMBL3191874 | — | — | 1 | 6.65 |
| CHEMBL1587116 | — | — | 1 | 6.64 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | 4.0 | 1 | 6.61 |
| CHEMBL1498488 | — | — | 1 | 6.59 |
| CHEMBL1595169 | — | — | 1 | 6.57 |
| CHEMBL1363437 | — | — | 1 | 6.53 |
| CHEMBL453974 | — | — | 1 | 6.51 |
| CHEMBL1329221 | — | — | 1 | 6.48 |
| CHEMBL1582760 | — | — | 1 | 6.47 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | -1.0 | 1 | 6.46 |
| CHEMBL1520346 | — | — | 1 | 6.46 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | 4.0 | 1 | 6.46 |
| CHEMBL587994 | — | — | 1 | 6.45 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | 4.0 | 1 | 6.43 |
| CHEMBL3196518 | — | — | 1 | 6.42 |
| CHEMBL1876078 | — | — | 1 | 6.42 |
| CHEMBL1350192 | — | — | 1 | 6.35 |
| CHEMBL1324197 | — | — | 1 | 6.33 |
| CHEMBL3182775 | — | — | 1 | 6.32 |
| CHEMBL1371056 | — | — | 1 | 6.32 |
| CHEMBL1580075 | — | — | 1 | 6.29 |
| CHEMBL1970422 | — | — | 1 | 6.27 |
| CHEMBL1998716 | — | — | 1 | 6.25 |
| CHEMBL1452795 | — | — | 1 | 6.23 |
| CHEMBL1424468 | — | — | 1 | 6.23 |
| CHEMBL1586371 | — | — | 1 | 6.23 |
| CHEMBL1459468 | — | — | 1 | 6.22 |
| CHEMBL1997171 | — | — | 1 | 6.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL323668 | — | EC50 | = | 126.0 | nM | 6.90 |
| CHEMBL225071 | RALTITREXED | EC50 | = | 192.0 | nM | 6.72 |
| CHEMBL3191874 | — | EC50 | = | 223.0 | nM | 6.65 |
| CHEMBL1587116 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1607 | TOPOTECAN HYDROCHLORIDE | EC50 | = | 246.0 | nM | 6.61 |
| CHEMBL1498488 | — | EC50 | = | 254.0 | nM | 6.59 |
| CHEMBL1595169 | — | EC50 | = | 272.0 | nM | 6.57 |
| CHEMBL1363437 | — | EC50 | = | 298.0 | nM | 6.53 |
| CHEMBL453974 | — | EC50 | = | 309.0 | nM | 6.51 |
| CHEMBL1329221 | — | EC50 | = | 334.0 | nM | 6.48 |
| CHEMBL1582760 | — | EC50 | = | 341.0 | nM | 6.47 |
| CHEMBL1520346 | — | EC50 | = | 345.0 | nM | 6.46 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | EC50 | = | 345.0 | nM | 6.46 |
| CHEMBL1200563 | CERIVASTATIN SODIUM | EC50 | = | 347.0 | nM | 6.46 |
| CHEMBL587994 | — | EC50 | = | 352.0 | nM | 6.45 |
| CHEMBL1200976 | IDARUBICIN HYDROCHLORIDE | EC50 | = | 371.0 | nM | 6.43 |
| CHEMBL1876078 | — | EC50 | = | 380.0 | nM | 6.42 |
| CHEMBL3196518 | — | EC50 | = | 382.0 | nM | 6.42 |
| CHEMBL1350192 | — | EC50 | = | 450.0 | nM | 6.35 |
| CHEMBL1324197 | — | EC50 | = | 469.0 | nM | 6.33 |
| CHEMBL3182775 | — | EC50 | = | 476.0 | nM | 6.32 |
| CHEMBL1371056 | — | EC50 | = | 479.0 | nM | 6.32 |
| CHEMBL1580075 | — | EC50 | = | 515.0 | nM | 6.29 |
| CHEMBL1970422 | — | EC50 | = | 538.0 | nM | 6.27 |
| CHEMBL1998716 | — | EC50 | = | 568.0 | nM | 6.25 |
| CHEMBL1452795 | — | EC50 | = | 587.0 | nM | 6.23 |
| CHEMBL1586371 | — | EC50 | = | 594.0 | nM | 6.23 |
| CHEMBL1424468 | — | EC50 | = | 594.0 | nM | 6.23 |
| CHEMBL917 | FLOXURIDINE | EC50 | = | 596.0 | nM | 6.22 |
| CHEMBL1459468 | — | EC50 | = | 607.0 | nM | 6.22 |
| CHEMBL1997171 | — | EC50 | = | 605.0 | nM | 6.22 |
| CHEMBL1500188 | — | EC50 | = | 609.0 | nM | 6.21 |
| CHEMBL1483593 | — | EC50 | = | 637.0 | nM | 6.20 |
| CHEMBL1405453 | — | EC50 | = | 632.0 | nM | 6.20 |
| CHEMBL1544633 | — | EC50 | = | 635.0 | nM | 6.20 |
| CHEMBL87 | — | EC50 | = | 627.0 | nM | 6.20 |
| CHEMBL1576251 | — | EC50 | = | 659.0 | nM | 6.18 |
| CHEMBL1393195 | — | EC50 | = | 667.0 | nM | 6.18 |
| CHEMBL1518905 | — | EC50 | = | 664.0 | nM | 6.18 |
| CHEMBL1545099 | — | EC50 | = | 668.0 | nM | 6.17 |
| CHEMBL1564670 | — | EC50 | = | 672.0 | nM | 6.17 |
| CHEMBL1462074 | — | EC50 | = | 676.0 | nM | 6.17 |
| CHEMBL1362687 | — | EC50 | = | 699.0 | nM | 6.16 |
| CHEMBL1611614 | — | EC50 | = | 702.0 | nM | 6.15 |
| CHEMBL1358722 | — | EC50 | = | 708.0 | nM | 6.15 |
| CHEMBL3199311 | — | EC50 | = | 712.0 | nM | 6.15 |
| CHEMBL1424118 | — | EC50 | = | 717.0 | nM | 6.14 |
| CHEMBL1467533 | — | EC50 | = | 745.0 | nM | 6.13 |
| CHEMBL1405749 | — | EC50 | = | 751.0 | nM | 6.12 |
| CHEMBL1399388 | — | EC50 | = | 769.0 | nM | 6.11 |